# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3774537 | 54k | INH | 0 | ALA3776421 | Not Active | % | Rattus norvegicus | ||||
2. | ALA4207014 | 19 | INH | = | 0 | % | ALA4191171 | % | Rattus norvegicus | |||
3. | ALA4177303 | ARC-1527 | Activity | = | 96.5 | % | ALA4157928 | % | Rattus norvegicus | |||
4. | ALA4279819 | (R)-6c | INH | = | 80 | % | ALA4258490 | % | Rattus norvegicus | |||
5. | ALA4224807 | 6 | INH | = | 80 | % | ALA4220902 | % | Rattus norvegicus | |||
6. | ALA3221816 | (R)-11d | IC50 | = | 519 | nM | ALA3226114 | 6.29 | nM | Rattus norvegicus | ||
7. | (3S)-N-[2-(3-hydroxypropoxy)-4-(1H-pyrazol-4-yl)phenyl]-6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide | (S)-11d | IC50 | < | 4 | nM | ALA3226114 | nM | Rattus norvegicus | |||
8. | ALA3221814 | (R)-11c | IC50 | = | 900 | nM | ALA3226114 | 6.05 | nM | Rattus norvegicus | ||
9. | ALA3221813 | (S)-11c | IC50 | < | 4 | nM | ALA3226114 | nM | Rattus norvegicus | |||
10. | ALA3221812 | (R)-11b | IC50 | = | 32 | nM | ALA3226114 | 7.50 | nM | Rattus norvegicus | ||
11. | ALA3221811 | (S)-11b | IC50 | < | 4 | nM | ALA3226114 | nM | Rattus norvegicus | |||
12. | ALA3221810 | (R)-11a | IC50 | = | 411 | nM | ALA3226114 | 6.39 | nM | Rattus norvegicus | ||
13. | ALA3221809 | (S)-11a | IC50 | < | 4 | nM | ALA3226114 | nM | Rattus norvegicus | |||
14. | ALA3221808 | (R)-1 | IC50 | = | 43 | nM | ALA3226114 | 7.37 | nM | Rattus norvegicus | ||
15. | Chroman 1 | (S)-1 | IC50 | < | 4 | nM | ALA3226114 | nM | Rattus norvegicus | |||
16. | AT13148 | AT-13148 | INH | > | 80 | % | ALA4022198 | % | Rattus norvegicus | |||
17. | ALA1077604 | 5 | Activity | = | 64 | % | ALA3830967 | % | Rattus norvegicus | |||
18. | ALA3815046 | 42 | Activity | = | -80 | % | ALA3815727 | % | Rattus norvegicus | |||
19. | ALA3814140 | 40 | Activity | = | -65 | % | ALA3815727 | % | Rattus norvegicus | |||
20. | ALA3814340 | 16 | Activity | = | -93 | % | ALA3815727 | % | Rattus norvegicus |