| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  LY2109761 | 15d | Ki | = | 300 | nmol/L | ALA5234117 | 6.52 | nM | Homo sapiens | ||
| 2. |  ALA4538174 | EUB0000298 | Kd | = | 54 | nM | ALA5213610 | 7.27 | nM | Homo sapiens | ||
| 3. |  ALA5188399 | 1 | Activity | <= | 70 | % | ALA5155252 | % | Homo sapiens | |||
| 4. |  ALA4455633 | 13 | INH | 0 | ALA4406346 | Active | % | Homo sapiens | ||||
| 5. |  ALA4447308 | 3 | INH | 0 | ALA4406346 | Active | % | Homo sapiens | ||||
| 6. |  ALA4436648 | CVM-05-002 | INH | 0 | ALA4406346 | Active | % | Homo sapiens | ||||
| 7. | ALA4436648 | CVM-05-002 | Activity | 0 | ALA4406341 | Active | Homo sapiens | |||||
| 8. |  ALA4455923 | 48c | INH | < | 50 | % | ALA4405592 | % | Homo sapiens | |||
| 9. |  ALA4559936 | (+/-)-6 | Activity | = | 19 | % | ALA4391610 | % | Homo sapiens | |||
| 10. |  ALA4564973 | 50 | INH | = | 100 | % | ALA4389984 | % | Homo sapiens | |||
| 11. |  ALA4555459 | 43 | INH | = | 100 | % | ALA4389507 | % | Homo sapiens | |||
| 12. |  ALA4473365 | 7c | Activity | = | 82 | % | ALA4382788 | % | Homo sapiens | |||
| 13. |  ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379461 | nM | Homo sapiens | |||
| 14. |  ALA4459587 | DC-TEADin02 | INH | = | 9 | % | ALA4378978 | % | Homo sapiens | |||
| 15. |  CDK9-IN-7 | 21e | INH | = | 15 | % | ALA4377924 | % | Homo sapiens | |||
| 16. |  ALA4533719 | 11 | INH | 0 | ALA4376028 | Not Active | % | Homo sapiens | ||||
| 17. |  ALA4462318 | 19i | Kd(free) | = | 7.385 | uM | ALA4371430 | 5.13 | nM | Homo sapiens | ||
| 18. |  ALA4443828 | 19h | Kd(free) | = | 1.86 | uM | ALA4371430 | 5.73 | nM | Homo sapiens | ||
| 19. |  Dasatinib | 2, BMS-354825 | Activity | = | 50 | % | ALA4808022 | % | Homo sapiens | |||
| 20. |  ALA4855726 | B3 | Activity | > | 75 | % | ALA4808022 | % | Homo sapiens |
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