# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Barasertib (AZD1152-HQPA) | 34 | Kd | = | 240 | nM | ALA1908821 | 6.62 | nM | Homo sapiens | ||
2. | Barasertib (AZD1152-HQPA) | 34 | Kd | = | 140 | nM | ALA1908820 | 6.85 | nM | Homo sapiens | ||
3. | Barasertib (AZD1152-HQPA) | 34 | Kd | = | 120 | nM | ALA1908819 | 6.92 | nM | Homo sapiens | ||
4. | Barasertib (AZD1152-HQPA) | 34 | Kd | = | 80 | nM | ALA1908818 | 7.10 | nM | Homo sapiens | ||
5. | Sorafenib | 5 | Kd | = | 22 | nM | ALA1908821 | 7.66 | nM | Homo sapiens | ||
6. | Sorafenib | 5 | Kd | = | 39 | nM | ALA1908820 | 7.41 | nM | Homo sapiens | ||
7. | Sorafenib | 5 | Kd | = | 7.4 | nM | ALA1908819 | 8.13 | nM | Homo sapiens | ||
8. | Sorafenib | 5 | Kd | = | 13 | nM | ALA1908818 | 7.89 | nM | Homo sapiens | ||
9. | Nilotinib (AMN-107) | 38 | Kd | > | 10000 | nM | ALA1908821 | nM | Homo sapiens | |||
10. | Nilotinib (AMN-107) | 38 | Kd | > | 10000 | nM | ALA1908820 | nM | Homo sapiens | |||
11. | Nilotinib (AMN-107) | 38 | Kd | = | 1100 | nM | ALA1908819 | 5.96 | nM | Homo sapiens | ||
12. | Nilotinib (AMN-107) | 38 | Kd | = | 870 | nM | ALA1908818 | 6.06 | nM | Homo sapiens | ||
13. | GSK690693 | 3g, GSK-690693 | Kd | > | 10000 | nM | ALA1908821 | nM | Homo sapiens | |||
14. | GSK690693 | 3g, GSK-690693 | Kd | > | 10000 | nM | ALA1908820 | nM | Homo sapiens | |||
15. | GSK690693 | 3g, GSK-690693 | Kd | = | 1300 | nM | ALA1908819 | 5.89 | nM | Homo sapiens | ||
16. | GSK690693 | 3g, GSK-690693 | Kd | > | 10000 | nM | ALA1908818 | nM | Homo sapiens | |||
17. | Canertinib (CI-1033) | 18 | Kd | > | 10000 | nM | ALA1908821 | nM | Homo sapiens | |||
18. | Canertinib (CI-1033) | 18 | Kd | > | 10000 | nM | ALA1908820 | nM | Homo sapiens | |||
19. | Canertinib (CI-1033) | 18 | Kd | = | 840 | nM | ALA1908819 | 6.08 | nM | Homo sapiens | ||
20. | Canertinib (CI-1033) | 18 | Kd | = | 4200 | nM | ALA1908818 | 5.38 | nM | Homo sapiens |