| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA363743 | 1 | pKi | = | 5.7 | ALA5247028 | 5.70 | nM | Homo sapiens | |||
| 2. |  JNJ 10397049 | 9 | pKi | = | 5.5 | ALA5247028 | 5.50 | nM | Homo sapiens | |||
| 3. |  ALA5273790 | 51 | Ki | = | 96 | nM | ALA5244921 | 7.02 | nM | Homo sapiens | ||
| 4. |  ALA3235249 | 1 | Ki | = | 1 | nM | ALA5244921 | 9.00 | nM | Homo sapiens | ||
| 5. |  filorexant | FILOREXANT | Ki | = | 2.5 | nM | ALA5244921 | 8.60 | nM | Homo sapiens | ||
| 6. |  ALA3586412 | 4 | Ki | = | 150 | nM | ALA5244921 | 6.82 | nM | Homo sapiens | ||
| 7. |  ALA5174113 | (-)-38; 38b | Ki | = | 5.23 | nM | ALA5243959 | 8.28 | nM | Homo sapiens | ||
| 8. |  ALA5172765 | (+)-38 | Ki | = | 2.17 | nM | ALA5243959 | 8.66 | nM | Homo sapiens | ||
| 9. |  ALA5271252 | (+-)-20d | Emax | = | 54 | % | ALA5243957 | % | Homo sapiens | |||
| 10. |  ALA5275698 | 27d | Emax | = | 11.1 | % | ALA5243957 | % | Homo sapiens | |||
| 11. |  ALA5278013 | 20a | Emax | = | 30.1 | % | ALA5243957 | % | Homo sapiens | |||
| 12. |  ALA5282613 | 20b | Emax | = | 2.21 | % | ALA5243957 | % | Homo sapiens | |||
| 13. |  ALA5289437 | 30d | Emax | = | 2.81 | % | ALA5243957 | % | Homo sapiens | |||
| 14. |  ALA5270685 | (-)-20d | Emax | = | 4.31 | % | ALA5243957 | % | Homo sapiens | |||
| 15. | ALA5278013 | 20a | Emax | = | 5.07 | % | ALA5243957 | % | Homo sapiens | |||
| 16. |  ALA5287067 | 25d | Emax | = | 5.66 | % | ALA5243957 | % | Homo sapiens | |||
| 17. |  ALA5273739 | (+-)-28d | Emax | = | 23.6 | % | ALA5243957 | % | Homo sapiens | |||
| 18. |  ALA5275530 | 28a | Emax | = | 11.8 | % | ALA5243957 | % | Homo sapiens | |||
| 19. |  ALA5270624 | 28c | Emax | = | 3.71 | % | ALA5243957 | % | Homo sapiens | |||
| 20. |  ALA5276558 | 32d | Emax | = | 2.65 | % | ALA5243957 | % | Homo sapiens |
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