# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PHA-848125 | 28, PHA-848125 | Kd | = | 13.6 | nM | ALA5230687 | 7.87 | nM | Homo sapiens | ||
2. | ALA4067978 | Bosutinib isomer | Kd | = | 77.5 | nM | ALA5230687 | 7.11 | nM | Homo sapiens | ||
3. | Bosutinib Isomer 1, Free Base | 1 (SKI-606) | Kd | = | 43.7 | nM | ALA5230687 | 7.36 | nM | Homo sapiens | ||
4. | ALA4075828 | 2; PF-03814735 | Kd | = | 78.7 | nM | ALA5230687 | 7.10 | nM | Homo sapiens | ||
5. | ALA5272317 | 39 | IC50 | = | 22.32 | uM | ALA5230686 | 4.65 | nM | Homo sapiens | ||
6. | ALA4529533 | MK-1775 | IC50 | = | 6.9 | nM | ALA5230685 | 8.16 | nM | Homo sapiens | ||
7. | ALA5273914 | 15 | IC50 | = | 10.4 | nM | ALA5230685 | 7.98 | nM | Homo sapiens | ||
8. | ALA5285380 | 14 | IC50 | = | 1.7 | nM | ALA5230685 | 8.77 | nM | Homo sapiens | ||
9. | ALA5291046 | 13 | IC50 | = | 7.8 | nM | ALA5230685 | 8.11 | nM | Homo sapiens | ||
10. | ALA5283663 | 12 | IC50 | = | 4.7 | nM | ALA5230685 | 8.33 | nM | Homo sapiens | ||
11. | ALA4780868 | 43; CJM061 | IC50 | = | 27.8 | nM | ALA5230684 | 7.56 | nM | Homo sapiens | ||
12. | MK-1775 | SID103905025 | IC50 | = | 5.1 | nM | ALA5230683 | 8.29 | nM | Homo sapiens | ||
13. | PD0166285 | 9 | IC50 | = | 24 | nM | ALA5230681 | 7.62 | nM | Homo sapiens | ||
14. | ALA181017 | 60 | IC50 | = | 0.55 | uM | ALA5230681 | 6.26 | nM | Homo sapiens | ||
15. | ALA180821 | 62 | IC50 | = | 0.54 | uM | ALA5230681 | 6.27 | nM | Homo sapiens | ||
16. | ALA181095 | 46 | IC50 | = | 0.99 | uM | ALA5230681 | 6.00 | nM | Homo sapiens | ||
17. | ALA366922 | 55 | IC50 | = | 0.04 | uM | ALA5230681 | 7.40 | nM | Homo sapiens | ||
18. | ALA113070 | 72 | IC50 | = | 0.032 | uM | ALA5230681 | 7.50 | nM | Homo sapiens | ||
19. | ALA181285 | 47 | IC50 | = | 0.086 | uM | ALA5230681 | 7.07 | nM | Homo sapiens | ||
20. | ALA178758 | 42 | IC50 | = | 0.12 | uM | ALA5230681 | 6.92 | nM | Homo sapiens |