# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Ribociclib | RIBOCICLIB | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
2. | Filgotinib (GLPG0634) | SID174006711 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
3. | ALA3991933 | Sapanisertib | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
4. | GDC-0941 | 17, GDC-0941 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
5. | PF-3758309 | 1, PF-3758309 | Kd apparent | = | 1282 | nM | ALA3991632 | 5.89 | Active | nM | Homo sapiens | |
6. | ALA522892 | 5 | Kd apparent | = | 17364 | nM | ALA3991632 | 4.76 | Active | nM | Homo sapiens | |
7. | MLN2480 | SID174006384 | Kd apparent | = | 296 | nM | ALA3991632 | 6.53 | Active | nM | Homo sapiens | |
8. | Linifanib (ABT-869) | 17p, ABT-869 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
9. | ALA1950289 | 1, CC-930 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
10. | Temsirolimus (CCI-779, NSC 683864) | Temsirolimus | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
11. | CAL-101 | 74, GS-1101, CAL-101 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
12. | SCIO 469 hydrochloride | SCIO-469 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
13. | ALA3182444 | SID174006374 | Kd apparent | = | 11 | nM | ALA3991632 | 7.96 | Active | nM | Homo sapiens | |
14. | Pelitinib | EKB-569 | Kd apparent | = | 1193 | nM | ALA3991632 | 5.92 | Active | nM | Homo sapiens | |
15. | ALA1094408 | 49 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
16. | Fedratinib (SAR302503, TG101348) | 2, TG101348 | Kd apparent | = | 1727 | nM | ALA3991632 | 5.76 | Active | nM | Homo sapiens | |
17. | RGB-286638 | RGB-286638 | Kd apparent | = | 1235 | nM | ALA3991632 | 5.91 | Active | nM | Homo sapiens | |
18. | SGX-523 | SGX-523 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
19. | Sotrastaurin | 1 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens | ||
20. | ALA1091644 | OSI-906 | Kd apparent | > | 30000 | nM | ALA3991632 | Inactive | nM | Homo sapiens |