# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2322896 | 6a, (3S,4S)-6a | IC50 | = | 29 | uM | ALA2330922 | 4.54 | nM | Homo sapiens | ||
2. | ALA2322611 | 12a, (3S,4S)-12a | IC50 | > | 30 | uM | ALA2330922 | nM | Homo sapiens | |||
3. | ALA2322207 | (3S,5R)-12 | IC50 | > | 30 | uM | ALA2329600 | nM | Homo sapiens | |||
4. | ALA3403995 | 23 | IC50 | > | 30 | uM | ALA3406671 | nM | Homo sapiens | |||
5. | ALA3400435 | 23 | IC50 | > | 10 | uM | ALA3404891 | nM | Homo sapiens | |||
6. | ALA3318957 | 31 | IC50 | > | 30 | uM | ALA3365829 | nM | Homo sapiens | |||
7. | ALA94762 | 38 | IC50 | > | 0 | M | ALA680907 | nM | Homo sapiens | |||
8. | ALA3142274 | 54 | Inhibition | = | 0 | % | ALA680909 | % | Homo sapiens | |||
9. | ALA3142283 | 48 | Inhibition | = | 0 | % | ALA680909 | % | Homo sapiens | |||
10. | ALA430933 | 49 | Inhibition | = | 0 | % | ALA680909 | % | Homo sapiens | |||
11. | ALA3348538 | 47 | Inhibition | = | 0 | % | ALA680909 | % | Homo sapiens | |||
12. | ALA3142268 | 45 | Inhibition | = | 7 | % | ALA680909 | % | Homo sapiens | |||
13. | ALA3348552 | 43 | Inhibition | = | 0 | % | ALA680909 | % | Homo sapiens | |||
14. | ALA3348552 | 43 | Inhibition | = | 0 | % | ALA757029 | % | Homo sapiens | |||
15. | ALA3348542 | 53 | Inhibition | = | 0 | % | ALA680909 | % | Homo sapiens | |||
16. | Acetyl-NH-val-cyclohexyl-CH2[nch2choh]CH2-benzyl-val-NH-acetyl | 18 | IC50 | = | 1 | uM | ALA680908 | 6.00 | nM | Homo sapiens | ||
17. | (2S)-N-[(2S,3R)-1-cyclohexyl-4,4-difluoro-3-hydroxy-4-{[(2S)-2-methylbutyl]carbamoyl}butan-2-yl]-2-[(2S)-2-[(morpholine-4-sulfonyl)amino]-3-phenylpropanamido]pent-4-enamide | 2 | Ki | = | 13 | nM | ALA680910 | 7.89 | nM | Homo sapiens | ||
18. | ALA88526 | 10 | Ki | > | 4000 | nM | ALA680910 | nM | Homo sapiens | |||
19. | ALA84970 | 7 | Ki | = | 19 | nM | ALA680910 | 7.72 | nM | Homo sapiens | ||
20. | ALA418948 | 12 | Ki | = | 110 | nM | ALA680910 | 6.96 | nM | Homo sapiens |