# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Gambogic acid | 1, GA | IC50 | = | 1.47 | uM | ALA5241836 | 5.83 | nM | Homo sapiens | ||
2. | ALA1269107 | 6i | IC50 | = | 76 | nM | ALA5241832 | 7.12 | nM | Homo sapiens | ||
3. | ALA538616 | 8r | IC50 | = | 0.31 | uM | ALA5241832 | 6.51 | nM | Homo sapiens | ||
4. | ABT-199 (GDC-0199) | VENETOCLAX | Ki | = | 48 | nM | ALA5234933 | 7.32 | nM | Homo sapiens | ||
5. | ALA443684 | Scheme 4, 11 | Ki | <= | 1 | nM | ALA5234929 | nM | Homo sapiens | |||
6. | ALA591346 | 7l; ABT737 | Ki | <= | 1 | nM | ALA5234928 | nM | Homo sapiens | |||
7. | ALA5285186 | Apogossypolone | Ki | = | 660 | nM | ALA5234926 | 6.18 | nM | Homo sapiens | ||
8. | Sabutoclax | (R,-,R)-11, atropisoer | IC50 | = | 0.31 | uM | ALA5234920 | 6.51 | nM | Homo sapiens | ||
9. | ALA5278443 | 1a | Ki | = | 22.2 | nM | ALA5234916 | 7.65 | nM | Homo sapiens | ||
10. | ALA4465826 | Lead Bim | Ki | = | 0.08 | nM | ALA5234916 | 10.10 | nM | Homo sapiens | ||
11. | ALA5288359 | 5 | Ki | = | 3.56 | uM | ALA5232900 | 5.45 | nM | Homo sapiens | ||
12. | ALA4160782 | 29 | Ki | = | 5.01 | uM | ALA5232900 | 5.30 | nM | Homo sapiens | ||
13. | ALA5283389 | 17cd | Ki | = | 1.67 | uM | ALA5232900 | 5.78 | nM | Homo sapiens | ||
14. | ALA5269202 | 17bd | Ki | = | 1.91 | uM | ALA5232900 | 5.72 | nM | Homo sapiens | ||
15. | ALA5266814 | 6e-OH | Ki | = | 1.63 | uM | ALA5232900 | 5.79 | nM | Homo sapiens | ||
16. | ALA5272657 | 17ag | Ki | = | 17.9 | uM | ALA5232900 | 4.75 | nM | Homo sapiens | ||
17. | ALA5279726 | 17ac | Ki | = | 10.8 | uM | ALA5232900 | 4.97 | nM | Homo sapiens | ||
18. | ALA5270912 | 17ab | Ki | = | 43.1 | uM | ALA5232900 | 4.37 | nM | Homo sapiens | ||
19. | ALA5288183 | 17aa | Ki | = | 154 | uM | ALA5232900 | nM | Homo sapiens | |||
20. | ALA5266385 | 6e-OH-5 | Ki | = | 2.91 | uM | ALA5232900 | 5.54 | nM | Homo sapiens |