# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5307562 | Ki | > | 5 | uM | ALA5304900 | Not Active | nM | Homo sapiens | |||
2. | ABT-263 | Scheme 4, 11 | IC50 | = | 0.003 | uM | ALA3132072 | 8.48 | nM | Homo sapiens | ||
3. | ALA3126113 | 4 | IC50 | > | 30 | uM | ALA3132072 | nM | Homo sapiens | |||
4. | 4-(4-((4'-Chloro-4,4-dimethyl-3,4,5,6-tetrahydro-[1,1'-biphenyl]-2-yl)methyl)piperazin-1-yl)benzoic acid | 5 | IC50 | = | 22 | uM | ALA3132072 | 4.66 | nM | Homo sapiens | ||
5. | ALA3126115 | 6 | IC50 | = | 8 | uM | ALA3132072 | 5.10 | nM | Homo sapiens | ||
6. | ALA3126116 | 7 | IC50 | = | 0.15 | uM | ALA3132072 | 6.82 | nM | Homo sapiens | ||
7. | ALA3126117 | 8 | IC50 | = | 26 | uM | ALA3132072 | 4.58 | nM | Homo sapiens | ||
8. | ALA3126118 | 9 | IC50 | = | 0.007 | uM | ALA3132072 | 8.14 | nM | Homo sapiens | ||
9. | ALA3126119 | 10 | IC50 | = | 0.004 | uM | ALA3132072 | 8.36 | nM | Homo sapiens | ||
10. | ALA3126120 | 11 | IC50 | = | 0.004 | uM | ALA3132072 | 8.43 | nM | Homo sapiens | ||
11. | ALA3125475 | 39b | Kd | = | 4.9 | uM | ALA3131102 | 5.31 | nM | Homo sapiens | ||
12. | ALA3125476 | 41 | Kd | = | 6.9 | uM | ALA3131102 | 5.16 | nM | Homo sapiens | ||
13. | ALA3125475 | 39b | Kd | = | 2.1 | uM | ALA3131101 | 5.68 | nM | Homo sapiens | ||
14. | ALA3125476 | 41 | Kd | = | 4 | uM | ALA3131101 | 5.40 | nM | Homo sapiens | ||
15. | ALA371861 | 1 | Kd | = | 1.4 | uM | ALA3131101 | 5.85 | nM | Homo sapiens | ||
16. | ALA371861 | 1 | Kd | = | 0.9 | uM | ALA3131102 | 6.05 | nM | Homo sapiens | ||
17. | ALA3342191 | 9 | IC50 | 270 | nM | ALA4883618 | Not Active | nM | Homo sapiens | |||
18. | A-1155463 | 17, A-1155463 | IC50 | 0.55 | nM | ALA4883618 | Active | nM | Homo sapiens | |||
19. | ALA4551344 | EUB0000746 | IC50 | > | 25 | uM | ALA4883618 | Not Active | nM | Homo sapiens | ||
20. | ALA4228713 | 22 | IC50 | 753 | nM | ALA4883618 | Not Active | nM | Homo sapiens |