# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5271820 | 61 | Ki | = | 0.41 | uM | ALA5242704 | 6.39 | nM | Homo sapiens | ||
2. | ALA5280830 | 60 | Ki | = | 0.45 | uM | ALA5242704 | 6.35 | nM | Homo sapiens | ||
3. | Gambogic acid | 1, GA | IC50 | = | 0.122 | uM | ALA5241841 | 6.91 | nM | Homo sapiens | ||
4. | ALA1269107 | 6i | IC50 | = | 1.3 | uM | ALA5241841 | 5.89 | nM | Homo sapiens | ||
5. | Gambogic acid | 1, GA | IC5 | = | 1.21 | uM | ALA5241837 | uM | Homo sapiens | |||
6. | ALA1269107 | 6i | IC50 | = | 31 | nM | ALA5241833 | 7.51 | nM | Homo sapiens | ||
7. | ALA538616 | 8r | IC50 | = | 0.32 | uM | ALA5241833 | 6.50 | nM | Homo sapiens | ||
8. | ALA4530348 | Nap-1 | IC50 | = | 2.11 | uM | ALA5234941 | 5.68 | nM | Homo sapiens | ||
9. | ALA476730 | 23 | Kd | = | 36.1 | uM | ALA5234939 | 4.44 | nM | Homo sapiens | ||
10. | ALA4102399 | 8a | IC50 | = | 4.27 | uM | ALA5234938 | 5.37 | nM | Homo sapiens | ||
11. | ABT-199 (GDC-0199) | VENETOCLAX | Ki | < | 0.01 | nM | ALA5234931 | nM | Homo sapiens | |||
12. | ALA443684 | Scheme 4, 11 | Ki | <= | 1 | nM | ALA5234927 | nM | Homo sapiens | |||
13. | ALA591346 | 7l; ABT737 | Ki | <= | 1 | nM | ALA5234927 | nM | Homo sapiens | |||
14. | ALA5285186 | Apogossypolone | Ki | = | 35 | nM | ALA5234925 | 7.46 | nM | Homo sapiens | ||
15. | ALA551288 | 2, Apogossypol | EC50 | = | 2.8 | uM | ALA5234923 | 5.55 | nM | Homo sapiens | ||
16. | Sabutoclax | (R,-,R)-11, atropisoer | IC50 | = | 0.32 | uM | ALA5234919 | 6.50 | nM | Homo sapiens | ||
17. | AT-101 | Gossypol | Ki | = | 0.32 | uM | ALA5234918 | 6.50 | nM | Homo sapiens | ||
18. | ALA288542 | SID174007075 | IC50 | = | 9 | uM | ALA5234917 | 5.05 | nM | Homo sapiens | ||
19. | ALA5283370 | 1b | Ki | = | 9.48 | nM | ALA5234915 | 8.02 | nM | Homo sapiens | ||
20. | ALA4465826 | Lead Bim | Ki | = | 16.9 | nM | ALA5234915 | 7.77 | nM | Homo sapiens |