# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Sulbactam | 1 | MIC | = | 1.56 | ug ml-1 | ALA4377161 | ug.mL-1 | Staphylococcus aureus | |||
2. | ALA3914769 | 6a | INH | 0 | ALA3877838 | % | Staphylococcus aureus | |||||
3. | ALA4170126 | 12d | FICI | = | 0.2 | ALA4139274 | Staphylococcus aureus | |||||
4. | ALA4164703 | 5 | FICI | = | 0.2 | ALA4139274 | Staphylococcus aureus | |||||
5. | ALA4170126 | 12d | MIC | = | 0.9 | ug ml-1 | ALA4139270 | ug.mL-1 | Staphylococcus aureus | |||
6. | ALA4164703 | 5 | MIC | = | 0.8 | ug ml-1 | ALA4139270 | ug.mL-1 | Staphylococcus aureus | |||
7. | ALA4170126 | 12d | INH | 0 | ALA4139264 | Not Active | % | Staphylococcus aureus | ||||
8. | ALA4164703 | 5 | INH | 0 | ALA4139264 | Not Active | % | Staphylococcus aureus | ||||
9. | ALA4170126 | 12d | INH | 0 | ALA4139263 | Active | % | Staphylococcus aureus | ||||
10. | ALA4164703 | 5 | INH | 0 | ALA4139263 | Active | % | Staphylococcus aureus | ||||
11. | penicillin G | Benzylpenicillin | Kcat | = | 65 | /s | ALA986867 | /s | Staphylococcus aureus | |||
12. | ceftobiprole | BPR, ceftobiprole | Km | = | 78 | uM | ALA986867 | nM | Staphylococcus aureus | |||
13. | cefaloridine | cephaloridine | Km | = | 110 | uM | ALA986867 | nM | Staphylococcus aureus | |||
14. | penicillin G | Benzylpenicillin | Activity | = | 1500000 | % | ALA986865 | % | Staphylococcus aureus | |||
15. | penicillin G | Benzylpenicillin | Activity | = | 46000 | % | ALA986868 | % | Staphylococcus aureus | |||
16. | Ceftazidime | CAZ | Kcat/Km | = | 0 | /s/microM | ALA986866 | /s/microM | Staphylococcus aureus | |||
17. | Cefepime | 82(Cefepime) | Kcat/Km | = | 0 | /s/microM | ALA986866 | /s/microM | Staphylococcus aureus | |||
18. | ceftobiprole | BPR, ceftobiprole | Kcat/Km | = | 0 | /s/microM | ALA986866 | /s/microM | Staphylococcus aureus | |||
19. | Ceftazidime | CAZ | Kcat | = | 0 | /s | ALA986867 | /s | Staphylococcus aureus | |||
20. | cefaloridine | cephaloridine | Kcat/Km | = | 0.001 | /s/microM | ALA986866 | /s/microM | Staphylococcus aureus |