# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4579120 | 40; E40 | Activity | = | 9.4 | % | ALA4396168 | % | Homo sapiens | |||
2. | ALA4471059 | 19 | INH | = | -7 | % | ALA4368573 | % | Homo sapiens | |||
3. | Pemigatinib | PEMIGATINIB | INH | 0 | ALA4810227 | Not Active | % | Homo sapiens | ||||
4. | FR191413 | 47c | IC50 | = | 0.69 | nM | ALA4734030 | 9.16 | nM | Homo sapiens | ||
5. | ALA3774617 | 97 | IC50 | = | 0.36 | nM | ALA4734030 | 9.44 | nM | Homo sapiens | ||
6. | FR190997 | 19a | IC50 | = | 0.41 | nM | ALA4734030 | 9.39 | nM | Homo sapiens | ||
7. | ALA4793451 | 4j; MGS0274 | Activity | 0 | ALA4708753 | Not Active | Homo sapiens | |||||
8. | ALA334014 | 3 | Activity | 0 | ALA4708753 | Not Active | Homo sapiens | |||||
9. | ALA1189175 | 94 | IC50 | = | 0.26 | nM | ALA4362061 | 9.59 | nM | Homo sapiens | ||
10. | Remibrutinib (LOU064) | 25; LOU064 | Activity | 0 | ALA4358604 | Not Active | Homo sapiens | |||||
11. | Belzutifan | 2; PT2977 | Activity | 0 | ALA4312731 | Not Active | Homo sapiens | |||||
12. | ALA4570711 | 5 | INH | = | 33 | % | ALA4311142 | % | Homo sapiens | |||
13. | ALA4442234 | 4 | INH | = | 34 | % | ALA4311142 | % | Homo sapiens | |||
14. | ALA4528035 | 1 | INH | = | 36 | % | ALA4311140 | % | Homo sapiens | |||
15. | ALA4444021 | 2 | INH | = | 65 | % | ALA4311140 | % | Homo sapiens | |||
16. | ALA4474137 | 3 | INH | = | 41 | % | ALA4311140 | % | Homo sapiens | |||
17. | ALA4460189 | 6 | INH | = | 45 | % | ALA4311140 | % | Homo sapiens | |||
18. | CHDI 00390576 | 22 | INH | < | 25 | % | ALA4311099 | % | Homo sapiens | |||
19. | ALA4437833 | 16 | INH | < | 25 | % | ALA4311099 | % | Homo sapiens | |||
20. | ALA3958704 | 8a | INH | < | 20 | % | ALA4184466 | % | Homo sapiens |