| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1472 | TRH | EC50 | = | 0.001 | uM | ALA3602664 | 9.00 | nM | Mus musculus | ||
| 2. |  ALA3600450 | 12e, (2S)-Pip-L-His(2-isopropyl)-L-ProNH2 | EC50 | = | 1 | uM | ALA3602664 | 6.00 | nM | Mus musculus | ||
| 3. |  ALA3600449 | 12d, (2S)-Pip-L-His(2-propyl)-L-ProNH2 | EC50 | = | 0.94 | uM | ALA3602664 | 6.03 | nM | Mus musculus | ||
| 4. |  ALA3600448 | 12c, 3-Apyz-L-His(2-propyl)-L-ProNH2 | EC50 | = | 1.56 | uM | ALA3602664 | 5.81 | nM | Mus musculus | ||
| 5. |  ALA3600447 | 12b, 5-Mpyz-L-His(2-propyl)-L-ProNH2 | EC50 | = | 0.017 | uM | ALA3602664 | 7.77 | nM | Mus musculus | ||
| 6. |  ALA3600446 | 12a, 2-Pyz-L-His(2-propyl)-L-ProNH2 | EC50 | = | 0.15 | uM | ALA3602664 | 6.82 | nM | Mus musculus | ||
| 7. |  ALA3600445 | 8l, 2-Pyz-L-His(2,5-diiodo-1-benzyl)-L-ProNH2 | EC50 | = | 0.98 | uM | ALA3602664 | 6.01 | nM | Mus musculus | ||
| 8. |  ALA3600444 | 8k, 5-Mpyz-L-His(2,5-diiodo-1-benzyl)-L-ProNH2 | EC50 | = | 0.74 | uM | ALA3602664 | 6.13 | nM | Mus musculus | ||
| 9. |  ALA3601786 | 8j, 2-Pyz-L-His(2,5-diiodo-1-ethyl)-L-ProNH2 | EC50 | = | 7.21 | uM | ALA3602664 | 5.14 | nM | Mus musculus | ||
| 10. |  ALA3601785 | 8i, 2-Pyz-L-His(5-bromo-1-methyl)-L-ProNH2 | EC50 | = | 0.34 | uM | ALA3602664 | 6.47 | nM | Mus musculus | ||
| 11. |  ALA3601784 | 8h, 2-Pyz-L-His(2,5-diiodo)-L-ProNH2 | EC50 | = | 11.28 | uM | ALA3602664 | 4.95 | nM | Mus musculus | ||
| 12. |  ALA3601783 | 8g, 3-Apyz-L-His(2,5-dibromo)-L-ProNH2 | EC50 | = | 1.41 | uM | ALA3602664 | 5.85 | nM | Mus musculus | ||
| 13. |  ALA3601782 | 8f, 3-Apyz-L-His(5-bromo)-L-ProNH2 | EC50 | = | 0.287 | uM | ALA3602664 | 6.54 | nM | Mus musculus | ||
| 14. |  ALA3601781 | 8e, 5-Mpyz-L-His(5-bromo)-L-ProNH2 | EC50 | = | 0.498 | uM | ALA3602664 | 6.30 | nM | Mus musculus | ||
| 15. |  ALA3600451 | 8a, 2-Pyz-L-His(5-chloro)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602662 | nM | Mus musculus | |||
| 16. |  ALA3600452 | 8b, 2-Pyz-L-His(5-bromo)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602662 | nM | Mus musculus | |||
| 17. |  ALA3600453 | 8c, 2-Pyz-L-His(2,5-dibromo)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602662 | nM | Mus musculus | |||
| 18. |  ALA3600454 | 8d, 2-Mpyz-L-His(2,5-dibromo)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602662 | nM | Mus musculus | |||
| 19. | ALA3601781 | 8e, 5-Mpyz-L-His(5-bromo)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602662 | nM | Mus musculus | |||
| 20. | ALA3601782 | 8f, 3-Apyz-L-His(5-bromo)-L-ProNH2 | IC50 | > | 50 | uM | ALA3602662 | nM | Mus musculus |
The page will load shortly, Thanks for your patience!