| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5027251 | EUB0001559 | EC50 | > | 50 | uM | ALA5304891 | Not Active | nM | Homo sapiens | ||
| 2. |  ALA4475494 | 19 | EC50 | = | 5.6 | uM | ALA5304891 | 5.25 | Not Active | nM | Homo sapiens | |
| 3. |  BI-3812 | 44 | % Ctrl | = | 88 | % | ALA5304291 | Not Active | % | Homo sapiens | ||
| 4. |  BI-3802 | BI-3802 | % Ctrl | = | 99 | % | ALA5304188 | Not Active | % | Homo sapiens | ||
| 5. |  ALA3775576 | 18 | Activity | = | 4 | % | ALA3779057 | % | Homo sapiens | |||
| 6. |  ALA3774448 | 17 | INH | = | 3 | % | ALA3776517 | % | Homo sapiens | |||
| 7. |  ALA3775393 | 16 | INH | 0 | ALA3776516 | Not Active | % | Homo sapiens | ||||
| 8. |  ALA3774885 | 39 | Activity | = | -8 | % | ALA3779057 | % | Homo sapiens | |||
| 9. |  ALA3775317 | 31 | Activity | = | -37 | % | ALA3779057 | % | Homo sapiens | |||
| 10. |  ALA3758502 | 1 | INH | = | -1.4 | % | ALA3761278 | % | Homo sapiens | |||
| 11. |  ALA3745885 | 7ao; ON1231320 | IC50 | > | 10 | uM | ALA3750189 | nM | Homo sapiens | |||
| 12. |  ALA3746293 | 23 | INH | = | -3.6 | % | ALA3751061 | % | Homo sapiens | |||
| 13. |  A-971432 | 29; A-971432 | IC50 | > | 10 | uM | ALA3743940 | nM | Homo sapiens | |||
| 14. |  ALA3671311 | BDBM130912 | IC50 | = | 2.064 | nM | ALA3707732 | 8.69 | 263061 | nM | Homo sapiens | |
| 15. |  ALA3671309 | BDBM130910 | IC50 | = | 3.483 | nM | ALA3707732 | 8.46 | 263060 | nM | Homo sapiens | |
| 16. |  ALA1980995 | SID103905531 | IC50 | = | 1.182 | nM | ALA3707732 | 8.93 | 263059 | nM | Homo sapiens | |
| 17. |  ALA3628628 | 5 | INH | = | 4.41 | % | ALA3631503 | % | Homo sapiens | |||
| 18. |  ALA3628627 | 4 | INH | = | 61.49 | % | ALA3631503 | % | Homo sapiens | |||
| 19. |  ALA166031 | 3 | INH | = | 96.69 | % | ALA3631503 | % | Homo sapiens | |||
| 20. |  2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile | 11 | IC50 | = | 1.19 | mM | ALA3631845 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!