# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BIX 02565 | 24, BIX 02565, eutamer | IC50 | = | 139 | nM | ALA5213138 | 6.86 | nM | Homo sapiens | ||
2. | ALA5187271 | 29 | INH | = | 46 | % | ALA5157149 | % | Homo sapiens | |||
3. | ALA5169393 | 11 | INH | = | 98 | % | ALA5157082 | % | Homo sapiens | |||
4. | ALA5182980 | 4 | INH | = | 92 | % | ALA5157082 | % | Homo sapiens | |||
5. | ALA5196221 | 4ACP | INH | = | 19 | % | ALA5133776 | % | Homo sapiens | |||
6. | ALA5170855 | 17b | Activity | = | 8 | % | ALA5129166 | % | Homo sapiens | |||
7. | ALA4445335 | Roxyl-ZV-5J | INH | = | 17 | % | ALA4408086 | % | Homo sapiens | |||
8. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405528 | % | Homo sapiens | |||
9. | BMS-690514 | BMS-690514 | Kd | < | 225 | nM | ALA4394544 | nM | Homo sapiens | |||
10. | ALA4559936 | (+/-)-6 | Activity | = | 31 | % | ALA4391544 | % | Homo sapiens | |||
11. | ALA4564973 | 50 | INH | = | 98 | % | ALA4389918 | % | Homo sapiens | |||
12. | ALA4555459 | 43 | INH | = | 85 | % | ALA4389441 | % | Homo sapiens | |||
13. | ALA4473365 | 7c | Activity | = | 3.1 | % | ALA4382722 | % | Homo sapiens | |||
14. | ALA4438748 | 12j | IC50 | > | 10 | uM | ALA4379225 | nM | Homo sapiens | |||
15. | ALA4459587 | DC-TEADin02 | INH | = | -4 | % | ALA4378859 | % | Homo sapiens | |||
16. | CDK9-IN-7 | 21e | INH | = | -6 | % | ALA4377824 | % | Homo sapiens | |||
17. | Dasatinib | 2, BMS-354825 | Activity | > | 75 | % | ALA4807976 | % | Homo sapiens | |||
18. | ALA4855726 | B3 | Activity | > | 75 | % | ALA4807976 | % | Homo sapiens | |||
19. | ALA4867844 | C7 | Activity | > | 75 | % | ALA4807976 | % | Homo sapiens | |||
20. | ALA2348350 | 15u | Activity | = | 90 | % | ALA4806731 | % | Homo sapiens |