# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3798256 | 6a | Activity | = | 96 | % | ALA3802249 | % | Homo sapiens | |||
2. | ALA3797579 | 23 | INH | = | 2.1 | % | ALA3801254 | % | Homo sapiens | |||
3. | ALA3798257 | 9d | IC50 | > | 1000 | nM | ALA3802291 | nM | Homo sapiens | |||
4. | ALA3798631 | 6i | IC50 | > | 1000 | nM | ALA3802291 | nM | Homo sapiens | |||
5. | ALA3799585 | 15 | IC50 | > | 10 | uM | ALA3802279 | nM | Homo sapiens | |||
6. | DRAK2-IN-1 | 16 | IC50 | > | 10 | uM | ALA3802279 | nM | Homo sapiens | |||
7. | ALA513703 | 3 | IC50 | > | 10 | uM | ALA3802279 | nM | Homo sapiens | |||
8. | ALA3785951 | 33 | IC50 | > | 10 | uM | ALA3789970 | nM | Homo sapiens | |||
9. | ALA3786167 | 28 | IC50 | > | 10 | uM | ALA3789970 | nM | Homo sapiens | |||
10. | ALA3785500 | 3 | IC50 | > | 10 | uM | ALA3789970 | nM | Homo sapiens | |||
11. | ALA3787112 | 2 | IC50 | = | 0.76 | uM | ALA3789970 | 6.12 | nM | Homo sapiens | ||
12. | ALA3787614 | 17 | IC50 | > | 10 | uM | ALA3789970 | nM | Homo sapiens | |||
13. | ALA1614712 | 1; NVP-AEW541 | IC50 | > | 5.5 | uM | ALA3789970 | nM | Homo sapiens | |||
14. | ALA3604631 | 28a | IC50 | = | 6 | nM | ALA3791910 | 8.22 | nM | Homo sapiens | ||
15. | ALA3787103 | 42a | IC50 | = | 20 | nM | ALA3791910 | 7.70 | nM | Homo sapiens | ||
16. | ALA3786976 | 42b | IC50 | = | 6 | nM | ALA3791910 | 8.22 | nM | Homo sapiens | ||
17. | ALA3787422 | 42c | IC50 | = | 129 | nM | ALA3791910 | 6.89 | nM | Homo sapiens | ||
18. | ALA3786006 | 42n | IC50 | = | 22 | nM | ALA3791910 | 7.66 | nM | Homo sapiens | ||
19. | ALA3785999 | 42d | IC50 | = | 56 | nM | ALA3791910 | 7.25 | nM | Homo sapiens | ||
20. | ALA3785711 | 42e | IC50 | = | 3 | nM | ALA3791910 | 8.52 | nM | Homo sapiens |