| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  GSK 2250665A | 13 | pIC50 | = | 6.6 | ALA2446678 | 6.60 | nM | Homo sapiens | |||
| 2. |  ALA2425654 | 3 | INH | < | 50 | % | ALA2428985 | % | Homo sapiens | |||
| 3. |  ALA2425645 | 11 | INH | < | 50 | % | ALA2428985 | % | Homo sapiens | |||
| 4. |  ALA2425646 | 12 | INH | < | 50 | % | ALA2428985 | % | Homo sapiens | |||
| 5. |  ALA2402081 | 37 | INH | = | 2 | % | ALA2405490 | % | Homo sapiens | |||
| 6. |  ALA2333445 | 1 | Activity | = | 102 | % | ALA2352144 | % | Homo sapiens | |||
| 7. |  ALA2325940 | 42 | INH | > | 80 | % | ALA2329207 | % | Homo sapiens | |||
| 8. |  ALA2029436 | 2q | Activity | 0 | ALA2033679 | Active | Homo sapiens | |||||
| 9. |  ALA2012574 | 42, LDN-211898 | INH | = | 2 | % | ALA2014510 | % | Homo sapiens | |||
| 10. |  ALA4080797 | 35 | Activity | = | 100 | % | ALA4055141 | % | Homo sapiens | |||
| 11. |  ALA4096145 | 2 | Activity | = | 99 | % | ALA4055141 | % | Homo sapiens | |||
| 12. |  ALA4104658 | 8 | INH | = | 52 | % | ALA4053916 | % | Homo sapiens | |||
| 13. |  ALA111612 | 10a | % Control | 100 | % | ALA4879980 | Not Active | % | Homo sapiens | |||
| 14. |  ALA4526341 | EUB0000736 | % Control | 100 | % | ALA4879980 | Not Active | % | Homo sapiens | |||
| 15. |  ABT-100 | EUB0000289 | % Control | 93 | % | ALA4879980 | Not Active | % | Homo sapiens | |||
| 16. |  ALA3701197 | BDBM161028 | % Control | 100 | % | ALA4879980 | Not Active | % | Homo sapiens | |||
| 17. |  ALA3697701 | BDBM161012 | % Control | 89 | % | ALA4879980 | Not Active | % | Homo sapiens | |||
| 18. |  2-methyl-N-[2-({3-[2-(prop-2-enamido)acetamido]phenyl}amino)pyrimidin-5-yl]-5-[3-(trifluoromethyl)benzamido]benzamide | 38 | IC50 | = | 6.3 | nM | ALA3292444 | 8.20 | nM | Homo sapiens | ||
| 19. |  2-methyl-N-(2-{[3-(prop-2-enamido)phenyl]amino}pyrimidin-5-yl)-5-[3-(trifluoromethyl)benzamido]benzamide | 31 | IC50 | = | 8.2 | nM | ALA3292444 | 8.09 | nM | Homo sapiens | ||
| 20. |  ALA4584981 | EUB0000747 | % Control | 82 | % | ALA4879980 | Not Active | % | Homo sapiens |
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