# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3086536 | (S,S)-13b | INH | > | 50 | % | ALA3088379 | % | Homo sapiens | |||
2. | GSK 2250665A | 13 | pIC50 | = | 7.1 | ALA2446682 | 7.10 | nM | Homo sapiens | |||
3. | ALA2425654 | 3 | INH | < | 50 | % | ALA2428347 | % | Homo sapiens | |||
4. | ALA2425652 | 4 | INH | < | 50 | % | ALA2428347 | % | Homo sapiens | |||
5. | ALA2425649 | 8 | INH | < | 50 | % | ALA2428347 | % | Homo sapiens | |||
6. | ALA2425645 | 11 | INH | < | 50 | % | ALA2428347 | % | Homo sapiens | |||
7. | ALA2425644 | 13 | INH | < | 50 | % | ALA2428347 | % | Homo sapiens | |||
8. | ALA2425646 | 12 | INH | < | 50 | % | ALA2428347 | % | Homo sapiens | |||
9. | ALA2402081 | 37 | INH | = | 0 | % | ALA2405484 | % | Homo sapiens | |||
10. | ALA2348865 | 9a, CC214-1 | Activity | = | 83 | % | ALA2352804 | % | Homo sapiens | |||
11. | ALA2325940 | 42 | INH | > | 80 | % | ALA2329204 | % | Homo sapiens | |||
12. | ALA2029438 | 2s | Activity | 0 | ALA2033666 | Active | Homo sapiens | |||||
13. | ALA2017557 | 8 | IC50 | = | 440.9 | nM | ALA2020890 | 6.36 | nM | Homo sapiens | ||
14. | 3-[(2Z)-2-[5-(difluoromethyl)-1,2-dihydrothieno[3,2-c]pyrazol-3-ylidene]indol-6-yl]pentan-3-ol | 7 | IC50 | = | 77.5 | nM | ALA2020890 | 7.11 | nM | Homo sapiens | ||
15. | ALA2017555 | 6 | IC50 | = | 241.4 | nM | ALA2020890 | 6.62 | nM | Homo sapiens | ||
16. | ALA2017554 | 5 | IC50 | = | 55.7 | nM | ALA2020890 | 7.25 | nM | Homo sapiens | ||
17. | ALA2017553 | 4 | IC50 | = | 66.5 | nM | ALA2020890 | 7.18 | nM | Homo sapiens | ||
18. | ALA2017552 | 3 | IC50 | = | 73.8 | nM | ALA2020890 | 7.13 | nM | Homo sapiens | ||
19. | ALA2012574 | 42, LDN-211898 | INH | = | 8 | % | ALA2014516 | % | Homo sapiens | |||
20. | ALA4080797 | 35 | Activity | = | 100 | % | ALA4055271 | % | Homo sapiens |