# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4646784 | Table 2, R5C4 | EC50 | = | 6 | nM | ALA5244623 | 8.22 | nM | Homo sapiens | ||
2. | ALA5271268 | 133 | EC50 | = | 50 | nM | ALA5244618 | 7.30 | nM | Homo sapiens | ||
3. | ALA5280836 | 135; Bms-98118 | EC50 | = | 71 | nM | ALA5244582 | 7.15 | nM | Homo sapiens | ||
4. | ALA2385460 | 26, AM-5262 | Activity | 0 | ALA5240318 | Active | Homo sapiens | |||||
5. | TAK-875 | TAK-875 | FC | = | 500 | ALA5240317 | Homo sapiens | |||||
6. | ALA5285139 | 83 | FC | = | 2 | ALA5240317 | Homo sapiens | |||||
7. | ALA2385460 | 26, AM-5262 | Efficacy | = | -25 | % | ALA5240316 | % | Homo sapiens | |||
8. | ALA2385460 | 26, AM-5262 | Efficacy | = | -25 | % | ALA5240315 | % | Homo sapiens | |||
9. | ALA5285139 | 83 | Efficacy | = | 35 | % | ALA5240314 | % | Homo sapiens | |||
10. | ALA5285139 | 83 | FC | = | 10 | ALA5240313 | Homo sapiens | |||||
11. | TAK-875 | TAK-875 | EC50 | = | 7.7 | nM | ALA5240307 | 8.11 | nM | Homo sapiens | ||
12. | ALA2385460 | 26, AM-5262 | EC50 | = | 1.3 | nM | ALA5240307 | 8.89 | nM | Homo sapiens | ||
13. | GPR40/FFAR1 modulator 1 | 94 | EC50 | = | 6.5 | uM | ALA5240307 | 5.19 | nM | Homo sapiens | ||
14. | ALA5266696 | 94 | Emax | = | 99 | % | ALA5240301 | % | Homo sapiens | |||
15. | ALA5279736 | 93 | Emax | = | 42 | % | ALA5240301 | % | Homo sapiens | |||
16. | ALA5271725 | 92 | Emax | = | 92 | % | ALA5240301 | % | Homo sapiens | |||
17. | ALA5288340 | 91 | Emax | = | 91 | % | ALA5240301 | % | Homo sapiens | |||
18. | ALA5273852 | 90 | Emax | = | 73 | % | ALA5240301 | % | Homo sapiens | |||
19. | ALA5283726 | 89 | Emax | = | 98 | % | ALA5240301 | % | Homo sapiens | |||
20. | ALA5280599 | 88 | Emax | = | 66 | % | ALA5240301 | % | Homo sapiens |