| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5270781 | 38 | IC50 | > | 2 | uM | ALA5252053 | nM | Homo sapiens | |||
| 2. |  CX-4945 (Silmitasertib) | 25n | Kd | = | 0.38 | nM | ALA5251705 | 9.42 | nM | Homo sapiens | ||
| 3. |  ALA5191682 | 105 | IC50 | = | 5.4 | uM | ALA5228619 | 5.27 | nM | Homo sapiens | ||
| 4. |  TBB | 63 | INH | = | 99.8 | % | ALA5215104 | % | Homo sapiens | |||
| 5. | ALA5191682 | 105 | INH | = | 61.6 | % | ALA5215104 | % | Homo sapiens | |||
| 6. |  ALA5220214 | 104a | INH | = | 79 | % | ALA5215104 | % | Homo sapiens | |||
| 7. |  Onvansertib (NMS-P937) | 7g | IC50 | = | 826 | nM | ALA5213129 | 6.08 | nM | Homo sapiens | ||
| 8. |  BI 2536 | 1 | % of control | = | 103 | % | ALA5213532 | % | Homo sapiens | |||
| 9. | CX-4945 (Silmitasertib) | 25n | IC50 | = | 1 | nM | ALA5210317 | 9.00 | nM | Homo sapiens | ||
| 10. | CX-4945 (Silmitasertib) | 25n | IC50 | = | 100 | nM | ALA5209905 | 7.00 | nM | Homo sapiens | ||
| 11. |  BGT226 (NVP-BGT226) maleate | BGT-226 | Delta TM | = | 1.43 | C | ALA5209710 | C | Homo sapiens | |||
| 12. |  Barasertib (AZD1152-HQPA) | 34 | Delta TM | = | 0.06 | C | ALA5209710 | C | Homo sapiens | |||
| 13. |  AZD6482 | AZD-6482 | Delta TM | = | -0.12 | C | ALA5209710 | C | Homo sapiens | |||
| 14. |  ASP3026 | ASP-3026 | Delta TM | = | -0.41 | C | ALA5209710 | C | Homo sapiens | |||
| 15. |  TC ASK 10 | EUB0000623aCl | Delta TM | = | -0.34 | C | ALA5209710 | C | Homo sapiens | |||
| 16. |  AP26113 | AP26113 | Delta TM | = | 1.62 | C | ALA5209710 | C | Homo sapiens | |||
| 17. |  AIM-100 | 2 | Delta TM | = | -0.88 | C | ALA5209710 | C | Homo sapiens | |||
| 18. |  Selonsertib (GS-4997) | SELONSERTIB | Delta TM | = | 0.45 | C | ALA5209710 | C | Homo sapiens | |||
| 19. |  SB590885 | 33, SB-590885 | Delta TM | = | 0.15 | C | ALA5209710 | C | Homo sapiens | |||
| 20. |  Roscovitine (Seliciclib,CYC202) | Roscovitine | Delta TM | = | 0.45 | C | ALA5209710 | C | Homo sapiens |
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