# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PF 05105679 | 8, PF-05105679 | % of effect | = | 22 | % | ALA5214519 | % | Homo sapiens | |||
2. | [³H]hemicholinium-3 | hemicholinium-3 | IC50 | 0 | ALA5209597 | Inhibitor: Almost Complete Inhibition At A Concentration Of 10 Μm | Homo sapiens | |||||
3. | Choline chloride | IB | EC50 | = | 17 | uM | ALA5209597 | 4.77 | Substrate | nM | Homo sapiens | |
4. | CHDI 00390576 | 22 | INH | < | 25 | % | ALA4311077 | % | Homo sapiens | |||
5. | ALA4437833 | 16 | INH | < | 25 | % | ALA4311077 | % | Homo sapiens | |||
6. | ALA4217988 | 5; PF-06456384 | IC50 | = | 120 | nM | ALA4179923 | 6.92 | nM | Homo sapiens | ||
7. | ALA4217988 | 5; PF-06456384 | Ki | = | 68 | nM | ALA4179923 | 7.17 | nM | Homo sapiens | ||
8. | ALA4217988 | 5; PF-06456384 | INH | = | 99 | % | ALA4179758 | % | Homo sapiens | |||
9. | PF 04418948 | 15, PF-04418948 | % inhibition | 4 | % | ALA4886970 | Not Active | % | Homo sapiens | |||
10. | PQCA | 4i | % inhibition | 29 | % | ALA4882986 | Not Active | % | Homo sapiens | |||
11. | PF-04457845 | 23, PF-04457845 | % inhibition | 18 | % | ALA4883148 | Not Active | % | Homo sapiens | |||
12. | PF 05105679 | 8, PF-05105679 | % inhibition | 22 | % | ALA4883082 | Not Active | % | Homo sapiens | |||
13. | THPP-1 | THPP-1 | % inhibition | 9 | % | ALA4882986 | Not Active | % | Homo sapiens | |||
14. | PPTN | 2 | % inhibition | -13 | % | ALA4882986 | Not Active | % | Homo sapiens | |||
15. | MLi-2 | 1; MLi-2 | % inhibition | 18 | % | ALA4882986 | Not Active | % | Homo sapiens | |||
16. | ALA3417525 | 69, BI665915 | % Ctrl | 101 | % | ALA4881719 | Not Active | % | Homo sapiens | |||
17. | ALA3183609 | SID160644130 | IC50 | 0 | ALA3404114 | Not Determined | Homo sapiens | |||||
18. | ALA3401758 | 10u | IC50 | 0 | ALA3404114 | Not Determined | Homo sapiens | |||||
19. | ALA3301712 | 10t | IC50 | 0 | ALA3404114 | Not Determined | Homo sapiens | |||||
20. | ALA3301821 | 10s | IC50 | 0 | ALA3404114 | Not Determined | Homo sapiens |