# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Gambogic acid | 1, GA | IC50 | = | 2.02 | uM | ALA5241838 | 5.70 | nM | Homo sapiens | ||
2. | ABT-199 (GDC-0199) | VENETOCLAX | Ki | = | 245 | nM | ALA5234934 | 6.61 | nM | Homo sapiens | ||
3. | ALA443684 | Scheme 4, 11 | Ki | <= | 1 | nM | ALA5234930 | nM | Homo sapiens | |||
4. | ABT-199 (GDC-0199) | VENETOCLAX | Ki | = | 245 | nM | ALA5163774 | 6.61 | nM | Homo sapiens | ||
5. | 3-Chloro-1-(3,4-dichlorophenyl)-4-(4-methylpiperazin-1-yl)pyrrole-2,5-dione | 1 | Ki | = | 12.5 | uM | ALA5163774 | 4.90 | nM | Homo sapiens | ||
6. | ALA3417701 | 30b | Ki | > | 0.66 | uM | ALA3417964 | nM | Homo sapiens | |||
7. | A-1155463 | 17, A-1155463 | Ki | = | 19 | nM | ALA3382391 | 7.72 | nM | Homo sapiens | ||
8. | ABT-737 | 2, ABT-737 | Ki | <= | 1 | nM | ALA3364173 | nM | Homo sapiens | |||
9. | ABT-199 (GDC-0199) | VENETOCLAX | Ki | = | 245 | nM | ALA4052852 | 6.61 | nM | Homo sapiens | ||
10. | ABT-737 | 2, ABT-737 | Ki | < | 1 | nM | ALA4052838 | nM | Homo sapiens | |||
11. | ALA3265299 | 21 | Ki | = | 1.58 | uM | ALA3266889 | 5.80 | nM | Homo sapiens | ||
12. | ALA3265297 | 19 | Ki | = | 1.36 | uM | ALA3266889 | 5.87 | nM | Homo sapiens | ||
13. | ALA3265296 | 18 | Ki | = | 4.41 | uM | ALA3266889 | 5.36 | nM | Homo sapiens | ||
14. | ALA3265295 | 17 | Ki | = | 2.19 | uM | ALA3266889 | 5.66 | nM | Homo sapiens | ||
15. | ALA3265294 | 16 | Ki | = | 1.92 | uM | ALA3266889 | 5.72 | nM | Homo sapiens | ||
16. | UMI-77 | SID49732904 | Ki | = | 8.19 | uM | ALA3266889 | 5.09 | nM | Homo sapiens | ||
17. | ALA2030270 | 1, 15a, 11a ,PI-8182 | Ki | = | 37.53 | uM | ALA3266889 | 4.43 | nM | Homo sapiens | ||
18. | ALA443684 | Scheme 4, 11 | IC50 | = | 0.07 | uM | ALA4409526 | 7.16 | nM | Homo sapiens | ||
19. | ALA4474764 | 13 | IC50 | = | 4.37 | uM | ALA4409526 | 5.36 | nM | Homo sapiens | ||
20. | ALA4560892 | 12 | IC50 | = | 21 | uM | ALA4409526 | 4.68 | nM | Homo sapiens |