# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2425654 | 3 | INH | = | 93 | % | ALA2427808 | % | Homo sapiens | |||
2. | ALA2425652 | 4 | INH | = | 95 | % | ALA2427808 | % | Homo sapiens | |||
3. | ALA2425649 | 8 | INH | = | 64 | % | ALA2427808 | % | Homo sapiens | |||
4. | ALA2425645 | 11 | INH | < | 50 | % | ALA2427808 | % | Homo sapiens | |||
5. | ALA2425644 | 13 | INH | = | 96 | % | ALA2427808 | % | Homo sapiens | |||
6. | ALA2425628 | 24f | Kd | = | 0.88 | uM | ALA2429321 | 6.06 | nM | Homo sapiens | ||
7. | ALA2425628 | 24f | INH | > | 85 | % | ALA2427808 | % | Homo sapiens | |||
8. | ALA2425646 | 12 | INH | < | 50 | % | ALA2427808 | % | Homo sapiens | |||
9. | N-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methylphenyl]acetamide | 7b | Activity | = | 22 | % | ALA2410933 | % | Homo sapiens | |||
10. | ALA2402081 | 37 | INH | = | -3 | % | ALA2405306 | % | Homo sapiens | |||
11. | ALA1725279 | SP-600125 | INH | 0 | ALA2383368 | Active | % | Homo sapiens | ||||
12. | ALA2063926 | 17 | IC50 | < | 10 | uM | ALA2065144 | nM | Homo sapiens | |||
13. | ALA2063926 | 17 | INH | < | 15 | % | ALA2065114 | % | Homo sapiens | |||
14. | ALA2017253 | 47 | INH | = | 25 | % | ALA2065114 | % | Homo sapiens | |||
15. | ALA2348862 | 10b, CC214-2 | Activity | = | 94 | % | ALA2350839 | % | Homo sapiens | |||
16. | ALA2333445 | 1 | Activity | = | 97 | % | ALA2352127 | % | Homo sapiens | |||
17. | ALA2348862 | 10b, CC214-2 | Activity | = | 98 | % | ALA2352817 | % | Homo sapiens | |||
18. | ALA2348865 | 9a, CC214-1 | Activity | = | 98 | % | ALA2350839 | % | Homo sapiens | |||
19. | XL388 | 28, XL388 | IC50 | > | 10000 | nM | ALA2345756 | nM | Homo sapiens | |||
20. | Khk-IN-1 | 8 | IC50 | > | 40 | uM | ALA2019669 | nM | Homo sapiens |