# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2152768 | 3 | INH | = | 4.1 | % | ALA2156517 | % | Homo sapiens | |||
2. | Borussertib | EUB0000645a | % Inhibition | 0 | % | ALA4888173 | Not Active | % | Homo sapiens | |||
3. | BAY-091 | EUB0001564 | % inhibition | -10.68 | % | ALA4887844 | Not Active | % | Homo sapiens | |||
4. | BI 605906 | BI605906 | % Ctrl | 90 | % | ALA4887405 | Not Active | % | Homo sapiens | |||
5. | ALA4475494 | 19 | % Inhibition | 9 | % | ALA4885954 | Not Active | % | Homo sapiens | |||
6. | ALA4580220 | EUB0000311 | % residual kinase activity | 94 | % | ALA4884530 | Not Active | % | Homo sapiens | |||
7. | Skepinone-L | 2, Skepinone-L | % Residual activity with Skepinone-L | 82 | % | ALA4883886 | Not Active | % | Homo sapiens | |||
8. | MLI-2 | 1; MLi-2 | % Inhibition | 21.597 | % | ALA4882710 | Not Active | % | Homo sapiens | |||
9. | ALA3417525 | 69, BI665915 | % Ctrl | 91 | % | ALA4881939 | Not Active | % | Homo sapiens | |||
10. | BAY-885 | BAY-885; 41 | % residual kinase activity | 102 | % | ALA4881292 | Not Active | % | Homo sapiens | |||
11. | ALA3929963 | BDBM179364 | IC50 | < | 100 | nM | ALA3887229 | 326009 | nM | Homo sapiens | ||
12. | ALA3940583 | BDBM179363 | IC50 | < | 100 | nM | ALA3887229 | 326008 | nM | Homo sapiens | ||
13. | ALA4111009 | BDBM179362 | IC50 | < | 100 | nM | ALA3887229 | 326007 | nM | Homo sapiens | ||
14. | ALA3935058 | BDBM179361 | IC50 | = | 300 | nM | ALA3887229 | 6.52 | 326006 | nM | Homo sapiens | |
15. | ALA3941003 | BDBM179360 | IC50 | = | 300 | nM | ALA3887229 | 6.52 | 326005 | nM | Homo sapiens | |
16. | ALA3895022 | BDBM179359 | IC50 | = | 750 | nM | ALA3887229 | 6.12 | 326004 | nM | Homo sapiens | |
17. | ALA3966339 | BDBM179358 | IC50 | = | 300 | nM | ALA3887229 | 6.52 | 326003 | nM | Homo sapiens | |
18. | ALA3980012 | BDBM179357 | IC50 | < | 100 | nM | ALA3887229 | 326002 | nM | Homo sapiens | ||
19. | ALA3947636 | BDBM179356 | IC50 | < | 100 | nM | ALA3887229 | 326001 | nM | Homo sapiens | ||
20. | ALA3971930 | BDBM179355 | IC50 | = | 300 | nM | ALA3887229 | 6.52 | 326000 | nM | Homo sapiens |