# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | (-)-Epigallocatechin gallate | 1 | Activity | = | 57.23 | % | ALA3293245 | % | Mus musculus | |||
2. | ALA3287409 | 4 | Activity | = | 56.03 | % | ALA3293244 | % | Mus musculus | |||
3. | ALA2177904 | (S)-25 | IC50 | = | 68 | nM | ALA2187563 | 7.17 | nM | Mus musculus | ||
4. | AZD3839 | 27 | IC50 | = | 436 | nM | ALA2187563 | 6.36 | nM | Mus musculus | ||
5. | ALA2177909 | (S)-10 | IC50 | = | 204 | nM | ALA2187563 | 6.69 | nM | Mus musculus | ||
6. | AZD3839 | (S)-32 | IC50 | = | 51 | nM | ALA2187563 | 7.29 | nM | Mus musculus | ||
7. | ALA2177914 | (S)-16 | IC50 | = | 53 | nM | ALA2187563 | 7.28 | nM | Mus musculus | ||
8. | ALA2177917 | 35 | IC50 | = | 40 | nM | ALA2187563 | 7.40 | nM | Mus musculus | ||
9. | ALA2177919 | 37 | IC50 | = | 30 | nM | ALA2187563 | 7.52 | nM | Mus musculus | ||
10. | AZ-4217 | 3 | IC50 | = | 2.6 | nM | ALA2187563 | 8.59 | nM | Mus musculus | ||
11. | ALA2177304 | (R)-19 | IC50 | = | 3.4 | nM | ALA2187563 | 8.47 | nM | Mus musculus | ||
12. | ALA3634123 | 3R-6c | IC50 | = | 4.3 | nM | ALA3635179 | 8.37 | nM | Mus musculus | ||
13. | ALA2403769 | 14 | IC50 | = | 4.5 | nM | ALA3635179 | 8.35 | nM | Mus musculus | ||
14. | ALA3634122 | 3R-6a | IC50 | = | 7.4 | nM | ALA3635179 | 8.13 | nM | Mus musculus | ||
15. | atabecestat | BDBM210070 | IC50 | = | 9.7 | nM | ALA4811867 | 8.01 | nM | Mus musculus | ||
16. | ALA4458974 | 3a; DV2-103 | INH | 0 | ALA4308602 | Active | % | Mus musculus | ||||
17. | ALA4458974 | 3a; DV2-103 | INH | 0 | ALA4308601 | Active | % | Mus musculus | ||||
18. | ALA4561358 | 5f | INH | 0 | ALA4308601 | Active | % | Mus musculus | ||||
19. | ALA4532540 | 5b | INH | 0 | ALA4308601 | Active | % | Mus musculus | ||||
20. | ALA4458974 | 3a; DV2-103 | INH | 0 | ALA4308600 | Active | % | Mus musculus |