| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA1085745 | 3, Table1 | IC50 | > | 10 | uM | ALA2072825 | nM | Homo sapiens | |||
| 2. |  ALA608263 | 47 | IC50 | = | 20 | uM | ALA2072825 | 4.70 | nM | Homo sapiens | ||
| 3. |  ALA589136 | 33 | IC50 | = | 20 | uM | ALA2072825 | 4.70 | nM | Homo sapiens | ||
| 4. |  ALA589135 | 32 | IC50 | = | 1.4 | uM | ALA2072825 | 5.85 | nM | Homo sapiens | ||
| 5. |  LY2452473 | LY2452473 | CL | = | 18 | uL/min | ALA3531005 | uL/min | Homo sapiens | |||
| 6. | LY2452473 | LY2452473 | CL | = | 1.79 | uL/min | ALA3531000 | uL/min | Homo sapiens | |||
| 7. |  Boceprevir | 70 | Compound recovery | 0 | ALA3541894 | metabolite_not_detected | Homo sapiens | |||||
| 8. |  Amiodarone | Amiodarone | Drug metabolism | 0 | ALA3529117 | metabolite_detected | Homo sapiens | |||||
| 9. | Amiodarone | Amiodarone | Drug metabolism | 0 | ALA3529125 | metabolite_detected | Homo sapiens | |||||
| 10. |  ALA3526949 | M11-2 | Drug metabolism | 0 | ALA3529128 | metabolite_detected | Homo sapiens | |||||
| 11. |  ALA3526948 | M11-1 | Drug metabolism | 0 | ALA3529128 | metabolite_detected | Homo sapiens | |||||
| 12. | ALA3526949 | M11-2 | Drug metabolism | 0 | ALA3529129 | metabolite_detected | Homo sapiens | |||||
| 13. | ALA3526948 | M11-1 | Drug metabolism | 0 | ALA3529129 | metabolite_detected | Homo sapiens | |||||
| 14. | Amiodarone | Amiodarone | Drug metabolism | 0 | ALA3529130 | metabolite_detected | Homo sapiens | |||||
| 15. | Amiodarone | Amiodarone | Drug metabolism | 0 | ALA3530847 | metabolite_detected | Homo sapiens | |||||
| 16. |  Vorapaxar (MK-5348) | 4, SCH-530348 | Drug metabolism | 0 | ALA3535001 | metabolite_not_detected | Homo sapiens | |||||
| 17. |  Telmisartan | Telmisartan | IC50 | = | 0.42 | uM | ALA3541093 | 6.38 | nM | Homo sapiens | ||
| 18. |  Flunarizine | 53 | IC50 | = | 0.94 | uM | ALA3541093 | 6.03 | nM | Homo sapiens | ||
| 19. |  Amodiaquine | AMODIAQUINE | IC50 | = | 0.99 | uM | ALA3541093 | 6.00 | nM | Homo sapiens | ||
| 20. |  ALA1484 | nicardipine | IC50 | = | 1.69 | uM | ALA3541093 | 5.77 | nM | Homo sapiens |
The page will load shortly, Thanks for your patience!