| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA301982 | 1 | Ki | = | 0.045 | uM | ALA5233906 | 7.35 | nM | Homo sapiens | ||
| 2. |  ALA4785914 | 19 | IC50 | > | 10 | uM | ALA4731223 | nM | Homo sapiens | |||
| 3. |  PDK4-IN-1 hydrochloride | 8c | IC50 | > | 50 | uM | ALA4333067 | nM | Homo sapiens | |||
| 4. |  PT-2385 | (S)-10i | Drug metabolism | 0 | ALA4312551 | Metabolite_Notdetected | Homo sapiens | |||||
| 5. |  PF-05221304 | 38 | IC50 | > | 20 | uM | ALA4669899 | nM | Homo sapiens | |||
| 6. |  ALA3398252 | 2 | Drug metabolism | 0 | ALA3398976 | metabolite_notdetected | Homo sapiens | |||||
| 7. |  Raltegravir (MK-0518) | 1, raltegravir | Drug metabolism | 0 | ALA3398976 | metabolite_detected | Homo sapiens | |||||
| 8. | ALA3398252 | 2 | Activity | 0 | ALA3398990 | Not Active | Homo sapiens | |||||
| 9. | ALA3398252 | 2 | IC50 | > | 300 | uM | ALA3399067 | nM | Homo sapiens | |||
| 10. |  1-pheny-3-methyl-5-pyrazolone | Edaravone | Drug metabolism | 0 | ALA3541745 | metabolite_detected | Homo sapiens | |||||
| 11. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Km | = | 2384 | uM | ALA3532181 | nM | Homo sapiens | |||
| 12. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Vmax | = | 1769 | pmol/min/g | ALA3532182 | pmol/min/g | Homo sapiens | |||
| 13. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | CL | = | 0.7 | uL/min/g | ALA3532183 | mL.min-1.g-1 | Homo sapiens | |||
| 14. | 1-pheny-3-methyl-5-pyrazolone | Edaravone | Drug metabolism | 0 | ALA3535214 | metabolite_not_detected | Homo sapiens | |||||
| 15. |  Gemfibrozil | 101 | CL free | = | 10.4 | ml/min/g | ALA3539806 | mL.min-1.g-1 | Homo sapiens | |||
| 16. | Gemfibrozil | 101 | CL free | = | 3.39 | ml/min/g | ALA3539813 | mL.min-1.g-1 | Homo sapiens | |||
| 17. | Gemfibrozil | 101 | CL free | = | 0.492 | ml/min/g | ALA3538589 | mL.min-1.g-1 | Homo sapiens | |||
| 18. | Gemfibrozil | 101 | Ratio | = | 0.328 | ALA3538596 | Homo sapiens | |||||
| 19. | Gemfibrozil | 101 | Ratio | = | 0.048 | ALA3541186 | Homo sapiens | |||||
| 20. | Gemfibrozil | 101 | Ratio | = | 6.89 | ALA3541193 | Homo sapiens |
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