# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA4785914 | 19 | IC50 | > | 10 | uM | ALA4731217 | nM | Homo sapiens | |||
2. | ALA4453227 | 13 | Km | = | 5.5 | uM | ALA4312568 | nM | Homo sapiens | |||
3. | Belzutifan | 2; PT2977 | Km | = | 10 | uM | ALA4312568 | nM | Homo sapiens | |||
4. | ALA4467490 | 9 | Km | = | 12 | uM | ALA4312568 | nM | Homo sapiens | |||
5. | ALA4170809 | (1S,2S)-10l | Km | = | 15 | uM | ALA4312568 | nM | Homo sapiens | |||
6. | ALA4169671 | (1S,2R)-10k | Km | = | 15 | uM | ALA4312568 | nM | Homo sapiens | |||
7. | ALA4437382 | 6 | Km | = | 12 | uM | ALA4312568 | nM | Homo sapiens | |||
8. | PT-2385 | (S)-10i | Km | = | 11 | uM | ALA4312568 | nM | Homo sapiens | |||
9. | ALA4453227 | 13 | Vmax | = | 440 | pmol/min | ALA4312567 | pmol/min | Homo sapiens | |||
10. | Belzutifan | 2; PT2977 | Vmax | = | 4.7 | pmol/min | ALA4312567 | pmol/min | Homo sapiens | |||
11. | ALA4467490 | 9 | Vmax | = | 1.4 | pmol/min | ALA4312567 | pmol/min | Homo sapiens | |||
12. | ALA4170809 | (1S,2S)-10l | Vmax | = | 50 | pmol/min | ALA4312567 | pmol/min | Homo sapiens | |||
13. | ALA4169671 | (1S,2R)-10k | Vmax | = | 14 | pmol/min | ALA4312567 | pmol/min | Homo sapiens | |||
14. | ALA4437382 | 6 | Vmax | = | 3.8 | pmol/min | ALA4312567 | pmol/min | Homo sapiens | |||
15. | PT-2385 | (S)-10i | Vmax | = | 280 | pmol/min | ALA4312567 | pmol/min | Homo sapiens | |||
16. | ALA4453227 | 13 | Km | = | 15 | uM | ALA4312566 | nM | Homo sapiens | |||
17. | Belzutifan | 2; PT2977 | Km | = | 15 | uM | ALA4312566 | nM | Homo sapiens | |||
18. | ALA4467490 | 9 | Km | = | 130 | uM | ALA4312566 | nM | Homo sapiens | |||
19. | ALA4170809 | (1S,2S)-10l | Km | = | 26 | uM | ALA4312566 | nM | Homo sapiens | |||
20. | ALA4169671 | (1S,2R)-10k | Km | = | 28 | uM | ALA4312566 | nM | Homo sapiens |