# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | BAY 678 | 17, BAY-678 | IC50 | > | 30 | uM | ALA5213826 | nM | Homo sapiens | |||
2. | ALA4556207 | 22 | Activity | 0 | ALA4380425 | Active | Homo sapiens | |||||
3. | ALA4554739 | 21 | Activity | 0 | ALA4380425 | Active | Homo sapiens | |||||
4. | ALA4560112 | 20 | Activity | 0 | ALA4380425 | Active | Homo sapiens | |||||
5. | ALA4465306 | 19 | Activity | 0 | ALA4380425 | Active | Homo sapiens | |||||
6. | ALA4561218 | 16 | Activity | 0 | ALA4380425 | Active | Homo sapiens | |||||
7. | ALA4554739 | 21 | IC50 | = | 290 | nM | ALA4380424 | 6.54 | nM | Homo sapiens | ||
8. | ALA4560112 | 20 | IC50 | = | 33 | nM | ALA4380424 | 7.48 | nM | Homo sapiens | ||
9. | ALA4592765 | 17 | IC50 | = | 10 | nM | ALA4380424 | 8.00 | nM | Homo sapiens | ||
10. | ALA4592765 | 17 | INH | > | 90 | % | ALA4380423 | % | Homo sapiens | |||
11. | ALA4583320 | RETY-pNA | Kcat/Km | = | 3.2 | 10'4/M/s | ALA4380420 | 10'4/M/s | Homo sapiens | |||
12. | ALA4520063 | FTDY-pNA | Kcat/Km | = | 3.8 | 10'4/M/s | ALA4380420 | 10'4/M/s | Homo sapiens | |||
13. | ALA4454436 | RTTY-pNA | Kcat/Km | = | 3.4 | 10'4/M/s | ALA4380420 | 10'4/M/s | Homo sapiens | |||
14. | ALA4549498 | NleTDY-pNA | Kcat/Km | = | 4 | 10'4/M/s | ALA4380420 | 10'4/M/s | Homo sapiens | |||
15. | ALA4583320 | RETY-pNA | Kcat | = | 13 | 1/s | ALA4380419 | 1/s | Homo sapiens | |||
16. | ALA4520063 | FTDY-pNA | Kcat | = | 14 | 1/s | ALA4380419 | 1/s | Homo sapiens | |||
17. | ALA4454436 | RTTY-pNA | Kcat | = | 18 | 1/s | ALA4380419 | 1/s | Homo sapiens | |||
18. | ALA4549498 | NleTDY-pNA | Kcat | = | 22 | 1/s | ALA4380419 | 1/s | Homo sapiens | |||
19. | ALA4583320 | RETY-pNA | Km | = | 410 | uM | ALA4380410 | nM | Homo sapiens | |||
20. | ALA4520063 | FTDY-pNA | Km | = | 370 | uM | ALA4380410 | nM | Homo sapiens |