# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | RN486 | 29, RN486 | IC50 | = | 29.2 | nM | ALA2060654 | 7.54 | nM | |||
2. | ALA4530401 | EUB0000704 | IC50 | > | 10 | uM | ALA4882585 | Not Active | nM | |||
3. | ALA3685796 | BDBM124625 | IC50 | 38 | nM | ALA4882585 | Active | nM | ||||
4. | PDK4-IN-1 hydrochloride | 8c | INH | 0 | ALA4333086 | Dose-dependent effect | % | |||||
5. | PDK4-IN-1 hydrochloride | 8c | OD | = | 0.2 | ALA4333087 | ||||||
6. | PDK4-IN-1 hydrochloride | 8c | OD | = | 0.126 | ALA4333088 | ||||||
7. | ALA3715003 | E63 | Activity | = | 5.7 | % | ALA3721016 | % | ||||
8. | ALA3719167 | E65 | Activity | = | 8.8 | % | ALA3721016 | % | ||||
9. | ALA3719048 | B174 | Activity | = | 8 | % | ALA3721016 | % | ||||
10. | ALA3718301 | C115 | Activity | = | 20 | % | ALA3721016 | % | ||||
11. | ALA3719254 | B13 | Activity | = | 10 | % | ALA3721016 | % | ||||
12. | ALA3717433 | C131 | Activity | = | 10.2 | % | ALA3721016 | % | ||||
13. | ALA3715476 | C133 | Activity | = | 12.4 | % | ALA3721016 | % | ||||
14. | ALA3715460 | C157 | Activity | = | 4.8 | % | ALA3721016 | % | ||||
15. | ALA3719252 | E51 | Activity | = | 5 | % | ALA3721016 | % | ||||
16. | ALA3719062 | E57 | Activity | = | 8.3 | % | ALA3721016 | % | ||||
17. | ALA3717422 | E59 | Activity | = | 5.1 | % | ALA3721016 | % | ||||
18. | ALA5085021 | 2 | FC | = | 12 | ALA5041219 | ||||||
19. | ALA5085021 | 2 | Cmax | = | 400 | nM | ALA5041218 | nM | ||||
20. | Disodium Cromoglycate | Disodium Cromoglycate | INH | = | 75 | % | ALA3259172 | % |