# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PF-06840003 | 6; EOS200271; PF-06840003 | Activity | 0 | ALA4058857 | Active | Mus musculus | |||||
2. | ALA5270178 | 5 | IC50 | = | 20 | uM | ALA5262183 | 4.70 | nM | Mus musculus | ||
3. | ALA5282240 | 3 | IC50 | = | 20 | uM | ALA5262183 | 4.70 | nM | Mus musculus | ||
4. | ALA599343 | 5 | INH | = | 31 | % | ALA1066923 | % | Mus musculus | |||
5. | ALA599531 | 4 | INH | = | 0 | % | ALA1066923 | % | Mus musculus | |||
6. | ALA599532 | 3 | INH | = | 40 | % | ALA1066923 | % | Mus musculus | |||
7. | ALA589275 | 2 | INH | = | 0 | % | ALA1066923 | % | Mus musculus | |||
8. | ALA599343 | 5 | IC50 | > | 10 | ug ml-1 | ALA1066922 | ug.mL-1 | Mus musculus | |||
9. | ALA599531 | 4 | IC50 | > | 10 | ug ml-1 | ALA1066922 | ug.mL-1 | Mus musculus | |||
10. | ALA599532 | 3 | IC50 | > | 10 | ug ml-1 | ALA1066922 | ug.mL-1 | Mus musculus | |||
11. | ALA589275 | 2 | IC50 | > | 10 | ug ml-1 | ALA1066922 | ug.mL-1 | Mus musculus | |||
12. | ALA550961 | 1 | IC50 | = | 8.3 | ug ml-1 | ALA1066922 | ug.mL-1 | Mus musculus | |||
13. | ALA599343 | 5 | INH | = | 44 | % | ALA1066919 | % | Mus musculus | |||
14. | ALA589275 | 2 | INH | = | 40 | % | ALA1066919 | % | Mus musculus | |||
15. | ALA599531 | 4 | INH | = | 40 | % | ALA1066919 | % | Mus musculus | |||
16. | ALA599343 | 5 | IC50 | = | 1 | ug ml-1 | ALA1066918 | ug.mL-1 | Mus musculus | |||
17. | ALA599531 | 4 | IC50 | > | 1 | ug ml-1 | ALA1066918 | ug.mL-1 | Mus musculus | |||
18. | ALA599532 | 3 | IC50 | = | 0.78 | ug ml-1 | ALA1066918 | ug.mL-1 | Mus musculus | |||
19. | ALA589275 | 2 | IC50 | > | 1 | ug ml-1 | ALA1066918 | ug.mL-1 | Mus musculus | |||
20. | ALA550961 | 1 | IC50 | = | 0.78 | ug ml-1 | ALA1066918 | ug.mL-1 | Mus musculus |