# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Brensocatib | 30; AZD7986 | IC50 | > | 20 | uM | ALA3859659 | nM | Homo sapiens | |||
2. | ALA3640116 | BDBM100336 | % Ctrl | 98 | % | ALA4887709 | Not Active | % | Homo sapiens | |||
3. | ALA4588900 | EUB0001182 | % Inhibition of Control Values | 12.3 | % | ALA4882567 | % | Homo sapiens | ||||
4. | ALA2338554 | 1 | Activity | = | 100 | % | ALA2340937 | % | Homo sapiens | |||
5. | ALA1241348 | 29, BI 201335 | INH | = | 0 | % | ALA1677868 | % | Homo sapiens | |||
6. | ALA4754916 | 25 | IC50 | = | 7.13 | uM | ALA4686520 | 5.15 | nM | Homo sapiens | ||
7. | ALA4743093 | 20 | IC50 | = | 9.54 | uM | ALA4686520 | 5.02 | nM | Homo sapiens | ||
8. | ALA4744124 | 19 | IC50 | = | 13.6 | uM | ALA4686520 | 4.87 | nM | Homo sapiens | ||
9. | ALA4752735 | 10 | IC50 | = | 12.4 | uM | ALA4686520 | 4.91 | nM | Homo sapiens | ||
10. | ALA1331625 | SID14736084 | IC50 | = | 11.8 | uM | ALA4686520 | 4.93 | nM | Homo sapiens | ||
11. | ALA4798763 | Z9 | IC50 | = | 11.5 | uM | ALA4686520 | 4.94 | nM | Homo sapiens | ||
12. | ALA4794067 | 54 | Activity | = | 85 | % | ALA4686519 | % | Homo sapiens | |||
13. | ALA4759795 | 53 | Activity | = | 60 | % | ALA4686519 | % | Homo sapiens | |||
14. | ALA4762267 | 52 | Activity | = | 63 | % | ALA4686519 | % | Homo sapiens | |||
15. | ALA4785867 | 51 | Activity | = | 69 | % | ALA4686519 | % | Homo sapiens | |||
16. | ALA4778457 | 50 | Activity | = | 73 | % | ALA4686519 | % | Homo sapiens | |||
17. | ALA4797796 | 49 | Activity | = | 100 | % | ALA4686519 | % | Homo sapiens | |||
18. | ALA4747196 | 48 | Activity | = | 80 | % | ALA4686519 | % | Homo sapiens | |||
19. | ALA4761185 | 47 | Activity | = | 92 | % | ALA4686519 | % | Homo sapiens | |||
20. | ALA4786943 | 46 | Activity | = | 41 | % | ALA4686519 | % | Homo sapiens |