# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | TG 003 | K00243, TG003 | IC50 | = | 12 | nM | ALA5116212 | 7.92 | nM | Mus musculus | ||
2. | ALA4442374 | 2-1k | INH | 0 | ALA4344352 | Active | % | Mus musculus | ||||
3. | ALA4550946 | 2-1l | INH | 0 | ALA4344352 | Active | % | Mus musculus | ||||
4. | 4-(7-methoxy-1-methylpyrido[3,4-b]indol-9-yl)butanamide | 2-2c | INH | 0 | ALA4344352 | Active | % | Mus musculus | ||||
5. | ALA4563765 | 2-2d | INH | 0 | ALA4344352 | Active | % | Mus musculus | ||||
6. | ALA4575812 | 2-2f | INH | 0 | ALA4344352 | Active | % | Mus musculus | ||||
7. | ALA269538 | 1 | INH | 0 | ALA4344352 | Active | % | Mus musculus | ||||
8. | leucettine L41 | L41 | Kd(free) | = | 0.065 | uM | ALA2186697 | 7.19 | nM | Mus musculus | ||
9. | leucettine L41 | L41 | Activity | 0 | ALA2186690 | Active | Mus musculus | |||||
10. | leucettine L41 | L41 | Activity | 0 | ALA2186681 | Active | Mus musculus | |||||
11. | leucettine L41 | L41 | INH | 0 | ALA2186261 | Dose-dependent effect | % | Mus musculus | ||||
12. | leucettine L41 | L41 | INH | 0 | ALA2183886 | Active | % | Mus musculus | ||||
13. | Alsterpaullone | 28d | INH | 0 | ALA2183886 | Not Active | % | Mus musculus | ||||
14. | ALA3092862 | 3a | Activity | 0 | ALA3097745 | Active | Mus musculus | |||||
15. | (5Z)-2-[4-[2-[2-[2-(2-aminoethoxy)ethoxy]ethoxy]ethoxy]anilino]-5-(1,3-benzodioxol-5-ylmethylidene)-1H-imidazol-4-one | 3b | Activity | 0 | ALA3097745 | Active | Mus musculus | |||||
16. | ALA3092864 | 3c | Activity | 0 | ALA3097745 | Active | Mus musculus | |||||
17. | ALA81714 | 15 | IC50 | = | 4.5 | uM | ALA1106599 | 5.35 | nM | Mus musculus | ||
18. | ALA37139 | 22 | IC50 | = | 1.3 | uM | ALA1106599 | 5.89 | nM | Mus musculus | ||
19. | ALA211756 | 1 | IC50 | > | 50 | uM | ALA871428 | nM | Mus musculus | |||
20. | ALA211756 | 1 | Inhibition | = | 74 | % | ALA871429 | % | Mus musculus |