# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA301982 | 1 | Ki | = | 14.2 | uM | ALA5233912 | 4.85 | nM | Rattus norvegicus | ||
2. | ALA301982 | 1 | IC50 | = | 23.2 | uM | ALA5233911 | 4.63 | nM | Rattus norvegicus | ||
3. | ALA5182450 | GZ | Ki | = | 52.6 | uM | ALA5118022 | 4.28 | nM | Rattus norvegicus | ||
4. | (+)-Ketoconazole | SID144204227 | INH | 0 | ALA5118020 | Active | % | Rattus norvegicus | ||||
5. | ALA4288347 | 2; K-604 | Drug metabolism | 0 | ALA4725830 | Metabolite_Detected | Rattus norvegicus | |||||
6. | ALA4288347 | 2; K-604 | Drug metabolism | 0 | ALA4725829 | Metabolite_Detected | Rattus norvegicus | |||||
7. | ALA3527054 | (R)-sulindac | Drug metabolism | 0 | ALA3528179 | metabolite_not_detected | Rattus norvegicus | |||||
8. | ALA3527054 | (R)-sulindac | Drug metabolism | 0 | ALA3528173 | metabolite_not_detected | Rattus norvegicus | |||||
9. | ALA2105653 | SETILEUTON | Km | = | 2.2 | uM | ALA3530305 | nM | Rattus norvegicus | |||
10. | ALA3526875 | M5 | Drug metabolism | 0 | ALA3530300 | metabolite_detected | Rattus norvegicus | |||||
11. | ALA2105653 | SETILEUTON | Drug metabolism | 0 | ALA3530296 | metabolite_detected | Rattus norvegicus | |||||
12. | ALA1200689 | NITRIC OXIDE | mechanism based inhibition | 0 | ALA1908274 | Cytochrome P450 mechanistic inhibitor: PMID 9400024 | Rattus norvegicus | |||||
13. | Indomethacin | Indomethacin | mechanism based inhibition | 0 | ALA1908273 | Cytochrome P450 mechanistic inhibitor: PMID 1187510 | Rattus norvegicus |