| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 14.99 | ALA5304885 | Homo sapiens | |||||
| 2. | ALA5306285 | EUB0002235 | delta Tm | = | 1.055 | ALA5304885 | Not Active | Homo sapiens | ||||
| 3. |  ALA5308262 | EUB0002234 | delta Tm Staurosporine positive control | = | 14.99 | ALA5304781 | Homo sapiens | |||||
| 4. | ALA5308262 | EUB0002234 | delta Tm | = | 0.939 | ALA5304781 | Not Active | Homo sapiens | ||||
| 5. |  ALA5308250 | EUB0002186 | delta Tm Staurosporine positive control | = | 16.37 | ALA5304632 | Homo sapiens | |||||
| 6. | ALA5308250 | EUB0002186 | delta Tm | = | 0.033 | ALA5304632 | Not Active | Homo sapiens | ||||
| 7. |  ALA5306577 | EUB0002354 | delta Tm Staurosporine positive control | = | 16.37 | ALA5304533 | Homo sapiens | |||||
| 8. | ALA5306577 | EUB0002354 | delta Tm | = | -0.258 | ALA5304533 | Not Active | Homo sapiens | ||||
| 9. |  ALA3745885 | 7ao; ON1231320 | IC50 | > | 10 | uM | ALA3748182 | nM | Homo sapiens | |||
| 10. |  ALA3628628 | 5 | INH | = | 0.89 | % | ALA3630492 | % | Homo sapiens | |||
| 11. |  ALA3628627 | 4 | INH | = | 87.03 | % | ALA3630492 | % | Homo sapiens | |||
| 12. |  ALA166031 | 3 | INH | = | 99.77 | % | ALA3630492 | % | Homo sapiens | |||
| 13. |  ALA3623443 | 22d | INH | > | 90 | % | ALA3624241 | % | Homo sapiens | |||
| 14. |  Staurosporine | 1 (Staurosporine) | Kd | = | 5.5 | nM | ALA5252322 | 8.26 | nM | Homo sapiens | ||
| 15. |  ALA5271697 | 8a | INH | = | 26 | % | ALA5252311 | % | Homo sapiens | |||
| 16. | ALA5271697 | 8a | deltaTm | = | 3.8 | degrees C | ALA5252300 | degrees C | Homo sapiens | |||
| 17. |  ALA187139 | 47 | % of control | = | 21 | % | ALA5213627 | % | Homo sapiens | |||
| 18. |  ALA4518706 | EUB0000702 | % of control | = | 4.8 | % | ALA5213308 | % | Homo sapiens | |||
| 19. |  ALA4538174 | EUB0000298 | Kd | = | 30 | nM | ALA5213606 | 7.52 | nM | Homo sapiens | ||
| 20. |  Enzastaurin (LY317615) | 1e | Kd | = | 76 | nM | ALA5214803 | 7.12 | nM | Homo sapiens |
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