| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  N-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methylphenyl]acetamide | 7b | Activity | = | 22 | % | ALA2410939 | % | Homo sapiens | |||
| 2. | N-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methylphenyl]acetamide | 7b | IC50 | = | 70 | nM | ALA2410929 | 7.16 | nM | Homo sapiens | ||
| 3. |  ALA2402081 | 37 | INH | = | -1 | % | ALA2405153 | % | Homo sapiens | |||
| 4. |  ALA2397315 | 31d-2 | IC50 | = | 10 | uM | ALA2399035 | 5.00 | nM | Homo sapiens | ||
| 5. |  ALA2333445 | 1 | Activity | = | 100 | % | ALA2352471 | % | Homo sapiens | |||
| 6. |  ALA2348862 | 10b, CC214-2 | Activity | = | 95 | % | ALA2353139 | % | Homo sapiens | |||
| 7. | ALA2348862 | 10b, CC214-2 | Activity | = | 86 | % | ALA2353641 | % | Homo sapiens | |||
| 8. |  ALA2348865 | 9a, CC214-1 | Activity | = | 79 | % | ALA2353139 | % | Homo sapiens | |||
| 9. |  ALA574646 | 2, EF31 | INH | = | 48 | % | ALA2342679 | % | Homo sapiens | |||
| 10. |  ALA2336377 | 16e | Activity | = | 18 | % | ALA2345618 | % | Homo sapiens | |||
| 11. |  ALA2336379 | 16g | Activity | = | 11 | % | ALA2345618 | % | Homo sapiens | |||
| 12. |  ALA269538 | 1 | IC50 | = | 800 | nM | ALA2320041 | 6.10 | nM | Homo sapiens | ||
| 13. |  TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 94 | % | ALA2015005 | % | Homo sapiens | |||
| 14. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 97 | % | ALA2015849 | % | Homo sapiens | |||
| 15. |  ALA2012574 | 42, LDN-211898 | INH | = | 97 | % | ALA2014921 | % | Homo sapiens | |||
| 16. |  ALA3297832 | 4 | IC50 | = | 1.2 | uM | ALA3299314 | 5.92 | nM | Homo sapiens | ||
| 17. |  BAY-091 | EUB0001564 | % inhibition | 7.66 | % | ALA4887850 | Not Active | % | Homo sapiens | |||
| 18. |  BI 605906 | BI605906 | % Ctrl | 92 | % | ALA4887408 | Not Active | % | Homo sapiens | |||
| 19. |  ALA4475494 | 19 | % Inhibition | 2 | % | ALA4885957 | Not Active | % | Homo sapiens | |||
| 20. |  ALA4580220 | EUB0000311 | % residual kinase activity | 97 | % | ALA4884290 | Not Active | % | Homo sapiens |
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