| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  MRT00033659 | MRT00033659 | Activity | = | 42.42 | % | ALA2434611 | % | Homo sapiens | |||
| 2. | MRT00033659 | MRT00033659 | Activity | = | 71.96 | % | ALA2434224 | % | Homo sapiens | |||
| 3. |  ALA2430324 | MRT00055778 | Activity | = | 94.19 | % | ALA2434611 | % | Homo sapiens | |||
| 4. | ALA2430324 | MRT00055778 | Activity | = | 98.87 | % | ALA2434224 | % | Homo sapiens | |||
| 5. |  D4476 | K00219, D4476 | Activity | = | 80 | % | ALA2434611 | % | Homo sapiens | |||
| 6. |  ALA576349 | IC261 | Activity | = | 96 | % | ALA2434195 | % | Homo sapiens | |||
| 7. |  N-(5-Pyridin-3-yl-1H-pyrazolo[3,4-b]pyridin-3-yl)butyramide | 22 | Activity | = | 31 | % | ALA2434611 | % | Homo sapiens | |||
| 8. | N-(5-Pyridin-3-yl-1H-pyrazolo[3,4-b]pyridin-3-yl)butyramide | 22 | Activity | = | 72 | % | ALA2434224 | % | Homo sapiens | |||
| 9. |  N-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methylphenyl]acetamide | 7b | Activity | = | 29 | % | ALA2410937 | % | Homo sapiens | |||
| 10. | N-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methylphenyl]acetamide | 7b | IC50 | = | 40 | nM | ALA2410931 | 7.40 | nM | Homo sapiens | ||
| 11. |  ALA2402081 | 37 | INH | = | 12 | % | ALA2405106 | % | Homo sapiens | |||
| 12. |  ALA2333445 | 1 | Activity | = | 101 | % | ALA2352173 | % | Homo sapiens | |||
| 13. |  ALA2348865 | 9a, CC214-1 | Activity | = | 87 | % | ALA2352551 | % | Homo sapiens | |||
| 14. |  XL388 | 28, XL388 | IC50 | > | 10000 | nM | ALA2343915 | nM | Homo sapiens | |||
| 15. |  ALA2336377 | 16e | Activity | = | 8 | % | ALA2339744 | % | Homo sapiens | |||
| 16. |  ALA2336379 | 16g | Activity | = | 6 | % | ALA2339744 | % | Homo sapiens | |||
| 17. |  TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 89 | % | ALA2015134 | % | Homo sapiens | |||
| 18. | TAE684 (NVP-TAE684) | 12, NVP-TAE684 | Activity | = | 86 | % | ALA2016266 | % | Homo sapiens | |||
| 19. |  ALA2012574 | 42, LDN-211898 | INH | = | 53 | % | ALA2014931 | % | Homo sapiens | |||
| 20. |  ALA5306285 | EUB0002235 | delta Tm Staurosporine positive control | = | 6.377 | ALA5304880 | Homo sapiens |
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