# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | CX-4945 (Silmitasertib) | 25n | IC50 | = | 35 | nM | ALA5212838 | 7.46 | nM | Homo sapiens | ||
2. | ALA4538591 | 36; BAY-440 | IC50 | = | 1140 | nM | ALA5210415 | 5.94 | nM | Homo sapiens | ||
3. | BAY-985 | 34; BAY-985 | IC50 | = | 2 | nM | ALA5210410 | 8.70 | nM | Homo sapiens | ||
4. | ALA4538591 | 36; BAY-440 | IC50 | > | 27000 | nM | ALA5210156 | nM | Homo sapiens | |||
5. | BAY-985 | 34; BAY-985 | IC50 | = | 312 | nM | ALA5210151 | 6.51 | nM | Homo sapiens | ||
6. | BAY-985 | 34; BAY-985 | IC50 | = | 74 | nM | ALA5209991 | 7.13 | nM | Homo sapiens | ||
7. | ALA5200234 | 2e | INH | = | 0 | % | ALA5158997 | % | Homo sapiens | |||
8. | ALA5186128 | 2b | INH | = | 0 | % | ALA5158997 | % | Homo sapiens | |||
9. | ALA5185043 | 2a | INH | = | 0 | % | ALA5158997 | % | Homo sapiens | |||
10. | ALA5178711 | 26; CS12192 | IC50 | = | 162 | nM | ALA5150290 | 6.79 | nM | Homo sapiens | ||
11. | ALA5206946 | 19k; 12 | INH | = | 77 | % | ALA5145159 | % | Homo sapiens | |||
12. | ALA5206613 | 8o; CZw-124 | INH | = | 21 | % | ALA5139831 | % | Homo sapiens | |||
13. | BX-795 | BX-795 | IC50 | = | 6 | nM | ALA5131710 | 8.22 | nM | Homo sapiens | ||
14. | ALA5185001 | 24j | INH | < | 40 | % | ALA5115501 | % | Homo sapiens | |||
15. | ALA4458300 | 4 | Activity | = | 75 | % | ALA4414289 | % | Homo sapiens | |||
16. | ALA4445335 | Roxyl-ZV-5J | INH | = | 9 | % | ALA4408151 | % | Homo sapiens | |||
17. | ALA4455923 | 48c | INH | < | 50 | % | ALA4405588 | % | Homo sapiens | |||
18. | ALA4559936 | (+/-)-6 | Activity | = | 10 | % | ALA4391606 | % | Homo sapiens | |||
19. | ALA4564973 | 50 | INH | = | 81 | % | ALA4389980 | % | Homo sapiens | |||
20. | ALA4555459 | 43 | INH | = | 57 | % | ALA4389503 | % | Homo sapiens |