# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2088198 | 15 | Time | = | 131 | min | ALA2089592 | hr | Cavia porcellus | |||
2. | ALA2088197 | 14 | Time | = | 32.5 | min | ALA2089592 | hr | Cavia porcellus | |||
3. | [³H]darifenacin | Darifenacin | Time | = | 30 | min | ALA2089592 | hr | Cavia porcellus | |||
4. | ALA2088198 | 15 | IC50 | = | 240 | nM | ALA2091590 | 6.62 | nM | Cavia porcellus | ||
5. | ALA2088197 | 14 | IC50 | = | 3.9 | nM | ALA2091590 | 8.41 | nM | Cavia porcellus | ||
6. | isoprenaline | 2 | pEC50 | = | 7.54 | ALA2340159 | 7.54 | nM | Cavia porcellus | |||
7. | ALA2335408 | 11a | pEC50 | = | 8.47 | ALA2340159 | 8.47 | nM | Cavia porcellus | |||
8. | ALA2335409 | 11b | pEC50 | = | 8.55 | ALA2340159 | 8.55 | nM | Cavia porcellus | |||
9. | ALA2335410 | 11c | pEC50 | = | 8.71 | ALA2340159 | 8.71 | nM | Cavia porcellus | |||
10. | ALA2335411 | 11d | pEC50 | = | 8.5 | ALA2340159 | 8.50 | nM | Cavia porcellus | |||
11. | ALA2335412 | 17a | pEC50 | = | 9.19 | ALA2340159 | 9.19 | nM | Cavia porcellus | |||
12. | ALA2335413 | 17b | pEC50 | = | 9.17 | ALA2340159 | 9.17 | nM | Cavia porcellus | |||
13. | ALA2335414 | 17c | pEC50 | = | 9.08 | ALA2340159 | 9.08 | nM | Cavia porcellus | |||
14. | ALA2335415 | 17d | pEC50 | = | 9.2 | ALA2340159 | 9.20 | nM | Cavia porcellus | |||
15. | isoprenaline | 2 | Emax | = | 100 | % | ALA2340159 | % | Cavia porcellus | |||
16. | ALA2335408 | 11a | Emax | = | 100 | % | ALA2340159 | % | Cavia porcellus | |||
17. | ALA2335409 | 11b | Emax | = | 103 | % | ALA2340159 | % | Cavia porcellus | |||
18. | ALA2335410 | 11c | Emax | = | 103 | % | ALA2340159 | % | Cavia porcellus | |||
19. | ALA2335411 | 11d | Emax | = | 105 | % | ALA2340159 | % | Cavia porcellus | |||
20. | ALA2335412 | 17a | Emax | = | 102 | % | ALA2340159 | % | Cavia porcellus |