# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5184598 | 33 | pIC50 | = | 9.3 | ALA5129843 | 9.30 | nM | Cavia porcellus | |||
2. | ALA5184455 | 32 | pIC50 | = | 10 | ALA5129843 | 10.00 | nM | Cavia porcellus | |||
3. | ALA5208201 | 31 | pIC50 | = | 10.3 | ALA5129843 | 10.30 | nM | Cavia porcellus | |||
4. | ALA5200887 | 54 | pIC50 | = | 9.1 | ALA5129843 | 9.10 | nM | Cavia porcellus | |||
5. | ALA5193853 | 53 | pIC50 | = | 9.4 | ALA5129843 | 9.40 | nM | Cavia porcellus | |||
6. | ALA5208957 | 52 | pIC50 | = | 9.4 | ALA5129843 | 9.40 | nM | Cavia porcellus | |||
7. | 4-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]butyl 5-[[3-[(S)-[[(3R)-1-azabicyclo[2.2.2]octan-3-yl]oxycarbonylamino]-phenylmethyl]phenoxy]methyl]-1-methylpyrazole-3-carboxylate | 29 | pIC50 | = | 10.1 | ALA5129843 | 10.10 | nM | Cavia porcellus | |||
8. | ALA5190387 | 51 | pIC50 | = | 9.8 | ALA5129843 | 9.80 | nM | Cavia porcellus | |||
9. | ALA298285 | 3 | INH | 0 | ALA4416568 | Dose-dependent effect | % | Cavia porcellus | ||||
10. | ALA4438390 | 2 | INH | 0 | ALA4416568 | Dose-dependent effect | % | Cavia porcellus | ||||
11. | isoprenaline | 2 | EC50 | = | 7.9 | nM | ALA4416568 | 8.10 | nM | Cavia porcellus | ||
12. | ALA298285 | 3 | EC50 | = | 0.8 | uM | ALA4416568 | 6.10 | nM | Cavia porcellus | ||
13. | ALA4438390 | 2 | EC50 | = | 2.8 | uM | ALA4416568 | 5.55 | nM | Cavia porcellus | ||
14. | ALA4445289 | (R)-18c | Time | > | 12 | hr | ALA4340589 | hr | Cavia porcellus | |||
15. | ALA4473515 | 9g | Time | > | 12 | hr | ALA4340589 | hr | Cavia porcellus | |||
16. | Salmeterol | 10 | Time | > | 12 | hr | ALA4340589 | hr | Cavia porcellus | |||
17. | ALA4445289 | (R)-18c | Time | = | 1.9 | min | ALA4340588 | hr | Cavia porcellus | |||
18. | ALA4473515 | 9g | Time | = | 2.3 | min | ALA4340588 | hr | Cavia porcellus | |||
19. | Salmeterol | 10 | Time | = | 14.2 | min | ALA4340588 | hr | Cavia porcellus | |||
20. | isoprenaline | 2 | Time | = | 2.2 | min | ALA4340588 | hr | Cavia porcellus |