# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2036813 | 4 | EC50 | = | 0.22 | uM | ALA5243292 | 6.66 | nM | Homo sapiens | ||
2. | ALA5277000 | 130c | EC50 | = | 0.22 | uM | ALA5243292 | 6.66 | nM | Homo sapiens | ||
3. | ALA1672755 | 1 | EC50 | = | 0.22 | uM | ALA5243292 | 6.66 | nM | Homo sapiens | ||
4. | ALA5281556 | 130a | EC50 | = | 0.22 | uM | ALA5243292 | 6.66 | nM | Homo sapiens | ||
5. | ALA5284951 | 130g | EC50 | = | 0.22 | uM | ALA5243292 | 6.66 | nM | Homo sapiens | ||
6. | ALA5275861 | 130f | EC50 | = | 0.22 | uM | ALA5243292 | 6.66 | nM | Homo sapiens | ||
7. | ALA5270112 | 130d | EC50 | = | 0.22 | uM | ALA5243292 | 6.66 | nM | Homo sapiens | ||
8. | ALA5194648 | 76 | INH | 0 | ALA5142415 | NA | % | Homo sapiens | ||||
9. | ALA5180818 | 42 | INH | 0 | ALA5142415 | NA | % | Homo sapiens | ||||
10. | ALA5171669 | 4 | INH | 0 | ALA5142415 | NA | % | Homo sapiens | ||||
11. | ALA5180892 | 1 | INH | 0 | ALA5142415 | NA | % | Homo sapiens | ||||
12. | GLPG 0974 | 99, GLPG0974 | INH | 0 | ALA3382554 | Not Active | % | Homo sapiens | ||||
13. | GSK137647A | 8, GSK137647A | pIC50 | < | 4.5 | ALA3362663 | nM | Homo sapiens | ||||
14. | GSK137647A | 8, GSK137647A | pEC50 | < | 4.3 | ALA3362662 | nM | Homo sapiens | ||||
15. | GSK137647A | 8, GSK137647A | pEC50 | < | 4.5 | ALA3365223 | nM | Homo sapiens | ||||
16. | ALA4162307 | 10 | INH | < | 10 | % | ALA4158299 | % | Homo sapiens | |||
17. | ALA4162307 | 10 | Activity | < | 10 | % | ALA4158298 | % | Homo sapiens | |||
18. | TUG-1375 | 31; TUG-1375 | Activity | 0 | ALA4158164 | Not Active | Homo sapiens | |||||
19. | ALA3601003 | 8d | EC50 | > | 10 | uM | ALA3602372 | nM | Homo sapiens | |||
20. | ALA3601001 | 8b | EC50 | > | 10 | uM | ALA3602372 | nM | Homo sapiens |