# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2381282 | 28a, diastereomer | Activity | 0 | ALA2382524 | Not Active | Homo sapiens | |||||
2. | ALA2381285 | 30a, diastereomer | Activity | 0 | ALA2382524 | Not Active | Homo sapiens | |||||
3. | ALA2315528 | 40 | pEC50 | < | 5 | ALA2320491 | nM | Homo sapiens | ||||
4. | ALA3480577 | DDD01251909 | Mean fold stimulation | 1.25 | ALA4883373 | Homo sapiens | ||||||
5. | GLPG 0974 | 99, GLPG0974 | INH | 0 | ALA3383169 | Dose-dependent effect | % | Homo sapiens | ||||
6. | GLPG 0974 | 99, GLPG0974 | IC50 | = | 483 | nM | ALA3383169 | 6.32 | nM | Homo sapiens | ||
7. | GLPG 0974 | 99, GLPG0974 | IC50 | = | 9 | nM | ALA3382548 | 8.05 | nM | Homo sapiens | ||
8. | ALA3353540 | 98 | IC50 | = | 138 | nM | ALA3382548 | 6.86 | nM | Homo sapiens | ||
9. | ALA3353539 | 97 | IC50 | = | 116 | nM | ALA3382548 | 6.94 | nM | Homo sapiens | ||
10. | ALA3353538 | 96 | IC50 | = | 90 | nM | ALA3382548 | 7.05 | nM | Homo sapiens | ||
11. | ALA3353537 | 95 | IC50 | > | 10000 | nM | ALA3382548 | nM | Homo sapiens | |||
12. | ALA3353536 | 94 | IC50 | = | 261 | nM | ALA3382548 | 6.58 | nM | Homo sapiens | ||
13. | ALA3353535 | 93 | IC50 | = | 95 | nM | ALA3382548 | 7.02 | nM | Homo sapiens | ||
14. | ALA3353534 | 92 | IC50 | = | 40 | nM | ALA3382548 | 7.40 | nM | Homo sapiens | ||
15. | ALA3353533 | 91 | IC50 | = | 36 | nM | ALA3382548 | 7.44 | nM | Homo sapiens | ||
16. | ALA3353532 | 90 | IC50 | = | 48 | nM | ALA3382548 | 7.32 | nM | Homo sapiens | ||
17. | ALA3353531 | 89 | IC50 | = | 500 | nM | ALA3382548 | 6.30 | nM | Homo sapiens | ||
18. | ALA3353530 | 88 | IC50 | = | 57 | nM | ALA3382548 | 7.24 | nM | Homo sapiens | ||
19. | ALA3353529 | 87 | IC50 | = | 711 | nM | ALA3382548 | 6.15 | nM | Homo sapiens | ||
20. | ALA3353528 | 86 | IC50 | = | 156 | nM | ALA3382548 | 6.81 | nM | Homo sapiens |