# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Gemcitabine | Gemzar | Km | = | 2.15 | uM | ALA3538236 | nM | Homo sapiens | |||
2. | 2′,2′-Difluoro-2′-deoxyuridine | dFdU | CL | = | 0.027 | ml/min/mg | ALA3541984 | mL.min-1.g-1 | Homo sapiens | |||
3. | Cytosine β-D-arabinofuranoside | 2 | CL | = | 231.4 | ml/min/mg | ALA3538240 | mL.min-1.g-1 | Homo sapiens | |||
4. | Cytosine β-D-arabinofuranoside | 2 | Km | = | 3.04 | uM | ALA3538244 | nM | Homo sapiens | |||
5. | Gemcitabine | Gemzar | CL | = | 491.9 | ml/min/mg | ALA3541975 | mL.min-1.g-1 | Homo sapiens | |||
6. | Cytosine β-D-arabinofuranoside | 2 | Vmax | = | 706.5 | nmol/min/mg | ALA3538244 | nmol/min/mg | Homo sapiens | |||
7. | Gemcitabine | Gemzar | Vmax | = | 1057 | nmol/min/mg | ALA3538236 | nmol/min/mg | Homo sapiens | |||
8. | ALA2426573 | 36 | IC50 | = | 14.5 | nM | ALA3381704 | 7.84 | nM | Homo sapiens | ||
9. | ALA2426573 | 36 | Ki(app) | = | 0.8 | nM | ALA3381705 | 9.10 | nM | Homo sapiens | ||
10. | ALA2426573 | 36 | IC50 | = | 1.4 | nM | ALA3381706 | 8.85 | nM | Homo sapiens | ||
11. | ALA2426574 | 37 | IC50 | = | 14.1 | nM | ALA3381704 | 7.85 | nM | Homo sapiens | ||
12. | ALA2426574 | 37 | Ki(app) | = | 0.5 | nM | ALA3381705 | 9.30 | nM | Homo sapiens | ||
13. | ALA2426574 | 37 | IC50 | = | 4.9 | nM | ALA3381706 | 8.31 | nM | Homo sapiens | ||
14. | ALA3358091 | 3 | IC50 | = | 11.2 | nM | ALA3381704 | 7.95 | nM | Homo sapiens | ||
15. | ALA3358091 | 3 | Ki(app) | = | 1.8 | nM | ALA3381705 | 8.74 | nM | Homo sapiens | ||
16. | ALA3358091 | 3 | IC50 | = | 21.8 | nM | ALA3381706 | 7.66 | nM | Homo sapiens | ||
17. | ALA3358092 | 4 | IC50 | = | 754 | nM | ALA3381704 | 6.12 | nM | Homo sapiens | ||
18. | ALA3358092 | 4 | Ki(app) | = | 735 | nM | ALA3381705 | 6.13 | nM | Homo sapiens | ||
19. | ALA3358092 | 4 | IC50 | = | 395 | nM | ALA3381706 | 6.40 | nM | Homo sapiens | ||
20. | ALA2426568 | 31 | IC50 | = | 26.1 | nM | ALA3381704 | 7.58 | nM | Homo sapiens |