| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5184598 | 33 | pIC50 | = | 8.1 | ALA5129841 | 8.10 | nM | Cavia porcellus | |||
| 2. |  ALA5184455 | 32 | pIC50 | = | 10 | ALA5129841 | 10.00 | nM | Cavia porcellus | |||
| 3. |  ALA5208201 | 31 | pIC50 | = | 9.7 | ALA5129841 | 9.70 | nM | Cavia porcellus | |||
| 4. |  ALA5200887 | 54 | pIC50 | = | 8.7 | ALA5129841 | 8.70 | nM | Cavia porcellus | |||
| 5. |  ALA5193853 | 53 | pIC50 | = | 9.9 | ALA5129841 | 9.90 | nM | Cavia porcellus | |||
| 6. |  ALA5208957 | 52 | pIC50 | = | 9.4 | ALA5129841 | 9.40 | nM | Cavia porcellus | |||
| 7. |  4-[[(2R)-2-hydroxy-2-(8-hydroxy-2-oxo-1H-quinolin-5-yl)ethyl]amino]butyl 5-[[3-[(S)-[[(3R)-1-azabicyclo[2.2.2]octan-3-yl]oxycarbonylamino]-phenylmethyl]phenoxy]methyl]-1-methylpyrazole-3-carboxylate | 29 | pIC50 | = | 9.7 | ALA5129841 | 9.70 | nM | Cavia porcellus | |||
| 8. |  ALA5190387 | 51 | pIC50 | = | 9.3 | ALA5129841 | 9.30 | nM | Cavia porcellus | |||
| 9. |  ALA517712 | atropine | pA2 | = | 8.99 | ALA4122103 | 8.99 | nM | Cavia porcellus | |||
| 10. |  ALA4126145 | 13 | pKb | = | 5.78 | ALA4122100 | Cavia porcellus | |||||
| 11. | ALA4126145 | 13 | INH | 0 | ALA4122100 | Dose-dependent effect | % | Cavia porcellus | ||||
| 12. |  ALA4129589 | 11 | pKb | = | 6.39 | ALA4122100 | Cavia porcellus | |||||
| 13. | ALA4129589 | 11 | INH | 0 | ALA4122100 | Dose-dependent effect | % | Cavia porcellus | ||||
| 14. | ALA4126145 | 13 | Activity | 0 | ALA4122098 | Not Active | Cavia porcellus | |||||
| 15. | ALA4129589 | 11 | Activity | 0 | ALA4122098 | Not Active | Cavia porcellus | |||||
| 16. |  ALA3219042 | 15 | Time | > | 11 | hr | ALA3227051 | hr | Cavia porcellus | |||
| 17. | ALA3219042 | 15 | EC50 | = | 12 | nM | ALA3227050 | 7.92 | nM | Cavia porcellus | ||
| 18. |  ALA4540849 | 14 | pKb | = | 6.35 | ALA4433283 | Cavia porcellus | |||||
| 19. |  ALA4586133 | 16 | pKb | = | 6.16 | ALA4433283 | Cavia porcellus | |||||
| 20. | ALA517712 | atropine | pKb | = | 8.99 | ALA4433283 | Cavia porcellus |
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