# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5274024 | 41; NEO2734 | Kd | = | 31 | nM | ALA5241958 | 7.51 | nM | Homo sapiens | ||
2. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | -2 | degrees C | ALA5236404 | degrees C | Homo sapiens | |||
3. | ALA5267793 | 9d | deltaTm | = | -1.5 | degrees C | ALA5236404 | degrees C | Homo sapiens | |||
4. | ALA5220994 | 28 | INH | = | 97 | % | ALA5218019 | % | Homo sapiens | |||
5. | ALA5219177 | 29 | pIC50 | = | 9 | ALA5217995 | 9.00 | nM | Homo sapiens | |||
6. | ALA5220956 | 26 | pIC50 | = | 9.2 | ALA5217995 | 9.20 | nM | Homo sapiens | |||
7. | ALA5219712 | 2 | pIC50 | = | 8 | ALA5217994 | 8.00 | nM | Homo sapiens | |||
8. | ALA1700017 | SID85269223 | pIC50 | = | 6.8 | ALA5217994 | 6.80 | nM | Homo sapiens | |||
9. | ALA5220994 | 28 | pIC50 | = | 10.1 | ALA5217994 | 10.10 | nM | Homo sapiens | |||
10. | ALA5219667 | 27 | pIC50 | = | 9.7 | ALA5217994 | 9.70 | nM | Homo sapiens | |||
11. | ALA5220956 | 26 | pIC50 | = | 9.5 | ALA5217994 | 9.50 | nM | Homo sapiens | |||
12. | ALA5220732 | 25 | pIC50 | = | 9.6 | ALA5217994 | 9.60 | nM | Homo sapiens | |||
13. | ALA5220447 | 24 | pIC50 | = | 9.6 | ALA5217994 | 9.60 | nM | Homo sapiens | |||
14. | ALA5219157 | 23 | pIC50 | = | 9.9 | ALA5217994 | 9.90 | nM | Homo sapiens | |||
15. | ALA5221053 | 22 | pIC50 | = | 10 | ALA5217994 | 10.00 | nM | Homo sapiens | |||
16. | ALA5219030 | 21 | pIC50 | = | 9.8 | ALA5217994 | 9.80 | nM | Homo sapiens | |||
17. | ALA5219204 | 20 | pIC50 | = | 7.8 | ALA5217994 | 7.80 | nM | Homo sapiens | |||
18. | ALA5219693 | 19 | pIC50 | = | 9.8 | ALA5217994 | 9.80 | nM | Homo sapiens | |||
19. | ALA5219466 | 18 | pIC50 | = | 8.7 | ALA5217994 | 8.70 | nM | Homo sapiens | |||
20. | ALA5219472 | 17 | pIC50 | = | 7.7 | ALA5217994 | 7.70 | nM | Homo sapiens |