# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | 2,9-Bis(3-(dimethylamino)propyl)anthra[2,1,9-def:6,5,10-d'e'f']diisoquinoline-1,3,8,10(2H,9H)-tetraone | 1, TEL03 | INH | 0 | ALA3128861 | Not Active | % | Homo sapiens | ||||
2. | 2,9-Bis(3-(dimethylamino)propyl)anthra[2,1,9-def:6,5,10-d'e'f']diisoquinoline-1,3,8,10(2H,9H)-tetraone | 1, TEL03 | INH | 0 | ALA3129417 | Not Active | % | Homo sapiens | ||||
3. | 2,9-Bis(3-(dimethylamino)propyl)anthra[2,1,9-def:6,5,10-d'e'f']diisoquinoline-1,3,8,10(2H,9H)-tetraone | 1, TEL03 | INH | 0 | ALA3128862 | Not Active | % | Homo sapiens | ||||
4. | ALA4637208 | EUB0001113 | pKd | 4.5 | ALA4886891 | nM | Homo sapiens | |||||
5. | ALA4639128 | 62 | Kd | 5700 | nM | ALA4886844 | nM | Homo sapiens | ||||
6. | ALA4536197 | EUB0000326 | KD | 20000 | nM | ALA4886506 | Not Active | nM | Homo sapiens | |||
7. | ALA4536197 | EUB0000326 | IC50 | > | 10000 | nM | ALA4886504 | Not Active | nM | Homo sapiens | ||
8. | A 485 | A-485 | KD | 15 | nM | ALA4886506 | Active | nM | Homo sapiens | |||
9. | A 485 | A-485 | IC50 | 9.8 | nM | ALA4886504 | Active | nM | Homo sapiens | |||
10. | GSK620 | 1; 20 | pKd | 5.1 | ALA4885841 | nM | Homo sapiens | |||||
11. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885786 | nM | Homo sapiens | ||||
12. | ALA4648362 | EUB0001116 | pKd | 4.6 | ALA4885718 | nM | Homo sapiens | |||||
13. | ALA5195288 | 27 | pKd | = | 5.6 | ALA5157247 | 5.60 | nM | Homo sapiens | |||
14. | EML 425 | 7h | alphaKi | = | 5.7 | uM | ALA3424835 | uM | Homo sapiens | |||
15. | EML 425 | 7h | alphaKi | = | 6.8 | uM | ALA3424834 | uM | Homo sapiens | |||
16. | EML 425 | 7h | INH | 0 | ALA3424841 | Active | % | Homo sapiens | ||||
17. | EML 425 | 7h | INH | 0 | ALA3424840 | tde | % | Homo sapiens | ||||
18. | EML 425 | 7h | INH | 0 | ALA3424839 | tde | % | Homo sapiens | ||||
19. | EML 425 | 7h | Ki | = | 2 | uM | ALA3424835 | 5.70 | nM | Homo sapiens | ||
20. | EML 425 | 7h | Ki | = | 9.4 | uM | ALA3424834 | 5.03 | nM | Homo sapiens |