| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | -3 | degrees C | ALA5236407 | degrees C | Homo sapiens | |||
| 2. |  ALA5267793 | 9d | deltaTm | = | -1.5 | degrees C | ALA5236407 | degrees C | Homo sapiens | |||
| 3. |  ALA609728 | 2 | IC50 | = | 5 | uM | ALA5232438 | 5.30 | nM | Homo sapiens | ||
| 4. |  ALA5220994 | 28 | INH | 0 | ALA5218025 | NA | % | Homo sapiens | ||||
| 5. |  GSK 4027 | (R,R)-32; GSK4027 | IC50 | = | 40 | uM | ALA5214226 | 4.40 | nM | Homo sapiens | ||
| 6. |  ALA4780673 | EUB0000253b | IC50 | > | 10 | uM | ALA5214214 | nM | Homo sapiens | |||
| 7. | ALA4780673 | EUB0000253b | Kd | = | 74 | nM | ALA5214213 | 7.13 | nM | Homo sapiens | ||
| 8. | ALA4780673 | EUB0000253b | dTm | = | 1.53 | K | ALA5214212 | K | Homo sapiens | |||
| 9. | GSK 4027 | (R,R)-32; GSK4027 | Ki | = | 1.4 | nM | ALA5210548 | 8.85 | nM | Homo sapiens | ||
| 10. |  L-45 | 8; L-Moses | IC50 | = | 48 | nM | ALA5210519 | 7.32 | nM | Homo sapiens | ||
| 11. | GSK 4027 | (R,R)-32; GSK4027 | IC50 | = | 60 | nM | ALA5210249 | 7.22 | nM | Homo sapiens | ||
| 12. | L-45 | 8; L-Moses | IC50 | = | 660 | nM | ALA5210229 | 6.18 | nM | Homo sapiens | ||
| 13. |  ALA5204783 | 8m | deltaTm | = | 0.25 | degrees C | ALA5162536 | degrees C | Homo sapiens | |||
| 14. |  ALA5206088 | 8l; XY153 | deltaTm | = | 0 | degrees C | ALA5162536 | degrees C | Homo sapiens | |||
| 15. |  ALA5205742 | 8k | deltaTm | = | -1 | degrees C | ALA5162536 | degrees C | Homo sapiens | |||
| 16. |  ALA5178480 | 8j | deltaTm | = | -0.5 | degrees C | ALA5162536 | degrees C | Homo sapiens | |||
| 17. | (+)-JQ1 (DMSO solution) | (+)-JQ1 | deltaTm | = | -0.5 | degrees C | ALA5162536 | degrees C | Homo sapiens | |||
| 18. |  ALA5179520 | 9g; Y08284 | deltaTm | = | -0.6 | degrees C | ALA5156575 | degrees C | Homo sapiens | |||
| 19. |  ALA5204688 | 9d | deltaTm | = | -0.3 | degrees C | ALA5156575 | degrees C | Homo sapiens | |||
| 20. |  ALA5192803 | 9c | deltaTm | = | -0.6 | degrees C | ALA5156575 | degrees C | Homo sapiens |
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