# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA217676 | MB-3 | IC50 | = | 100 | uM | ALA4275278 | 4.00 | nM | Homo sapiens | ||
2. | ALA4637208 | EUB0001113 | pKd | 4.7 | ALA4886893 | nM | Homo sapiens | |||||
3. | ALA4639128 | 62 | Kd | 30000 | nM | ALA4886846 | nM | Homo sapiens | ||||
4. | A 485 | A-485 | % inhibition | -31.2 | % | ALA4886593 | Not Active | % | Homo sapiens | |||
5. | GSK620 | 1; 20 | pKd | 4.5 | ALA4885843 | nM | Homo sapiens | |||||
6. | GSK046 | 15; GSK046 | Kd | 30000 | nM | ALA4885788 | nM | Homo sapiens | ||||
7. | ALA4648362 | EUB0001116 | pKd | 4.5 | ALA4885720 | nM | Homo sapiens | |||||
8. | EML 425 | 7h | INH | 0 | ALA3424831 | Not Active | % | Homo sapiens | ||||
9. | GSK1324726A (I-BET726) | 45 | pIC50 | < | 6.5 | ALA3383425 | nM | Homo sapiens | ||||
10. | Butyrolactone 3 | 102 | IC50 | = | 100 | uM | ALA3391520 | 4.00 | nM | Homo sapiens | ||
11. | BAZ2-ICR | 13, BAZ2-ICR | Delta TM | = | 0.16 | C | ALA4650129 | C | Homo sapiens | |||
12. | TP-472 | 1; TP-472 | Delta TM | = | 0.61 | C | ALA4650129 | C | Homo sapiens | |||
13. | L-45 | 8; L-Moses | Delta TM | = | 3.75 | C | ALA4650129 | C | Homo sapiens | |||
14. | PFI-4 | 11 | Delta TM | = | 0.21 | C | ALA4650129 | C | Homo sapiens | |||
15. | I-BRD9 | 45; I-BRD9 | Delta TM | = | 1.26 | C | ALA4650129 | C | Homo sapiens | |||
16. | NVS-CECR2-1 | NVS-1 | Delta TM | = | 1.2 | C | ALA4650129 | C | Homo sapiens | |||
17. | ALA4650212 | EUB0000324a | Delta TM | = | -0.21 | C | ALA4650129 | C | Homo sapiens | |||
18. | OF 1 | 8 | Delta TM | = | 0.57 | C | ALA4650129 | C | Homo sapiens | |||
19. | NI-57 | 76; NI-57 | Delta TM | = | 0.45 | C | ALA4650129 | C | Homo sapiens | |||
20. | bromosporine | Bromosporine | Delta TM | = | 1.01 | C | ALA4650129 | C | Homo sapiens |