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# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3798741 | EPZ031686 | INH | < | 30 | % | ALA3803383 | % | Homo sapiens | |||
2. | ALA3798468 | EPZ030456 | INH | < | 30 | % | ALA3803383 | % | Homo sapiens | |||
3. | ALA3780926 | 7 | INH | 0 | ALA3784095 | Not Active | % | Homo sapiens | ||||
4. | cyproheptadine | 7 | IC50 | = | 20 | uM | ALA3626829 | 4.70 | nM | Homo sapiens | ||
5. | ALA3623770 | DC-S238 | IC50 | = | 4.88 | uM | ALA3626816 | 5.31 | nM | Homo sapiens | ||
6. | ALA3623769 | DC-S258 | IC50 | = | 61.55 | uM | ALA3626816 | 4.21 | nM | Homo sapiens | ||
7. | ALA3623753 | DC-S240 | IC50 | = | 49.52 | uM | ALA3626816 | 4.30 | nM | Homo sapiens | ||
8. | ALA3623752 | DC-S237 | IC50 | = | 37.67 | uM | ALA3626816 | 4.42 | nM | Homo sapiens | ||
9. | ALA3623751 | DC-S239 | IC50 | = | 4.59 | uM | ALA3626816 | 5.34 | nM | Homo sapiens | ||
10. | ALA3623592 | DC-S100 | IC50 | = | 30.04 | uM | ALA3626816 | 4.52 | nM | Homo sapiens | ||
11. | ALA1577117 | SID22413928 | IC50 | = | 61.75 | uM | ALA3626816 | 4.21 | nM | Homo sapiens | ||
12. | ALA3623579 | DC-S130 | IC50 | = | 189.7 | uM | ALA3626816 | nM | Homo sapiens | |||
13. | ALA3623578 | DC-S129 | IC50 | = | 89.18 | uM | ALA3626816 | 4.05 | nM | Homo sapiens | ||
14. | ALA3623770 | DC-S238 | INH | = | 94.71 | % | ALA3626815 | % | Homo sapiens | |||
15. | ALA3623769 | DC-S258 | INH | = | 70.44 | % | ALA3626815 | % | Homo sapiens | |||
16. | ALA3623768 | DC-S257 | INH | = | -2.55 | % | ALA3626815 | % | Homo sapiens | |||
17. | ALA3623767 | DC-S256 | INH | = | -5.57 | % | ALA3626815 | % | Homo sapiens | |||
18. | ALA3623766 | DC-S255 | INH | = | -6.45 | % | ALA3626815 | % | Homo sapiens | |||
19. | ALA3623765 | DC-S254 | INH | = | -7.88 | % | ALA3626815 | % | Homo sapiens | |||
20. | ALA3623764 | DC-S253 | INH | = | -4.7 | % | ALA3626815 | % | Homo sapiens |
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Standard Type
Target Type
Organism Taxonomy L1
Organism Taxonomy L2
Organism Taxonomy L3
Target Organism
Aladdin Value
BAO Label
- percent inhibition 216
- IC50 131
- fold activation 25
- percent activity 8
- Kd 4
- EC50 2
- Ki 2
- T1/2 1
- result 1
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