# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | Dorsomorphin | 1 | IC50 | = | 95 | nM | ALA5252283 | 7.02 | nM | Homo sapiens | ||
2. | ALA5273533 | 37 | IC50 | > | 1000 | nM | ALA5244434 | nM | Homo sapiens | |||
3. | ALA5281283 | 18 | IC50 | > | 1000 | nM | ALA5244434 | nM | Homo sapiens | |||
4. | TP0427736 HCl | 3a | IC50 | = | 836 | nmol/L | ALA5234113 | 6.08 | nM | Homo sapiens | ||
5. | PF-06952229 | PF-06952229 | IC50 | > | 1000 | uM | ALA5224850 | nM | Homo sapiens | |||
6. | ALA5202351 | (S)-31 | Activity | < | 1 | % | ALA5159144 | % | Homo sapiens | |||
7. | ALA5197985 | 12e | IC50 | 0 | ALA5133125 | ND | Homo sapiens | |||||
8. | ALA5194265 | 12d | IC50 | 0 | ALA5133125 | ND | Homo sapiens | |||||
9. | ALA5190190 | 12c | IC50 | 0 | ALA5133125 | ND | Homo sapiens | |||||
10. | ALA5175201 | 12b | IC50 | = | 400 | nM | ALA5133125 | 6.40 | nM | Homo sapiens | ||
11. | ALA5196379 | 12a, racemic mixture | IC50 | = | 2368 | nM | ALA5133125 | 5.63 | nM | Homo sapiens | ||
12. | ALA5200241 | 11i | IC50 | = | 161 | nM | ALA5133125 | 6.79 | nM | Homo sapiens | ||
13. | ALA5178564 | 11h | IC50 | = | 129 | nM | ALA5133125 | 6.89 | nM | Homo sapiens | ||
14. | ALA5186575 | 11g | IC50 | = | 171 | nM | ALA5133125 | 6.77 | nM | Homo sapiens | ||
15. | ALA5205781 | 11f, racemic mixture | IC50 | = | 186 | nM | ALA5133125 | 6.73 | nM | Homo sapiens | ||
16. | ALA5189461 | 11e | IC50 | = | 151 | nM | ALA5133125 | 6.82 | nM | Homo sapiens | ||
17. | ALA5195236 | 11d, racemic mixture | IC50 | = | 274 | nM | ALA5133125 | 6.56 | nM | Homo sapiens | ||
18. | ALA5207070 | 11c | IC50 | = | 193 | nM | ALA5133125 | 6.71 | nM | Homo sapiens | ||
19. | ALA5189688 | 11b | IC50 | = | 129 | nM | ALA5133125 | 6.89 | nM | Homo sapiens | ||
20. | ALA5183080 | 11a | IC50 | = | 161 | nM | ALA5133125 | 6.79 | nM | Homo sapiens |