# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3780032 | 5; IACS-4759 | INH | 0 | ALA3782142 | Not Active | % | Homo sapiens | ||||
2. | ALA3775317 | 31 | Activity | = | 21 | % | ALA3776645 | % | Homo sapiens | |||
3. | ALA3775576 | 18 | Activity | = | 33 | % | ALA3776645 | % | Homo sapiens | |||
4. | ALA3774885 | 39 | Activity | = | -7 | % | ALA3776645 | % | Homo sapiens | |||
5. | ALA3771285 | 12 | Activity | = | 100 | % | ALA3773976 | % | Homo sapiens | |||
6. | ALA3758502 | 1 | INH | = | 70.7 | % | ALA3762140 | % | Homo sapiens | |||
7. | ALA3746293 | 23 | INH | = | -3.9 | % | ALA3751271 | % | Homo sapiens | |||
8. | ALA3628628 | 5 | INH | = | -11.44 | % | ALA3631722 | % | Homo sapiens | |||
9. | ALA166031 | 3 | INH | = | -13.93 | % | ALA3631722 | % | Homo sapiens | |||
10. | ALA3628627 | 4 | INH | = | 42.36 | % | ALA3631722 | % | Homo sapiens | |||
11. | ALA3629616 | 1; Wrightiadione | Activity | = | 82 | % | ALA3630039 | % | Homo sapiens | |||
12. | 2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile | 11 | INH | = | 7.1 | % | ALA3631702 | % | Homo sapiens | |||
13. | PF-06952229 | PF-06952229 | IC50 | = | 0.057 | uM | ALA5224851 | 7.24 | nM | Homo sapiens | ||
14. | PF-06952229 | PF-06952229 | INH | > | 50 | % | ALA5224842 | % | Homo sapiens | |||
15. | ALA4750687 | EUB0000312b | IC50 | = | 126 | nM | ALA5210411 | 6.90 | nM | Homo sapiens | ||
16. | ALA4741904 | EUB0000710a | IC50 | > | 10000 | nM | ALA5210166 | nM | Homo sapiens | |||
17. | ALA4750687 | EUB0000312b | IC50 | = | 526 | nM | ALA5210152 | 6.28 | nM | Homo sapiens | ||
18. | ALA4741904 | EUB0000710a | EC50 | > | 10000 | nM | ALA5209999 | nM | Homo sapiens | |||
19. | ALA4750687 | EUB0000312b | EC50 | > | 1000 | nM | ALA5209992 | nM | Homo sapiens | |||
20. | ALA3298678 | 38 | INH | = | -2.5 | % | ALA3361853 | % | Homo sapiens |