# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | PF-06952229 | PF-06952229 | IC50 | = | 7.29 | uM | ALA5224855 | 5.14 | nM | Homo sapiens | ||
2. | ALA5205791 | 1 | IC50 | = | 45 | nM | ALA5133121 | 7.35 | nM | Homo sapiens | ||
3. | ALA5197985 | 12e | IC50 | = | 29 | nM | ALA5133121 | 7.54 | nM | Homo sapiens | ||
4. | ALA5194265 | 12d | IC50 | = | 164 | nM | ALA5133121 | 6.79 | nM | Homo sapiens | ||
5. | ALA5190190 | 12c | IC50 | = | 5764 | nM | ALA5133121 | 5.24 | nM | Homo sapiens | ||
6. | ALA5175201 | 12b | IC50 | = | 27 | nM | ALA5133121 | 7.57 | nM | Homo sapiens | ||
7. | ALA5196379 | 12a, racemic mixture | IC50 | = | 61 | nM | ALA5133121 | 7.21 | nM | Homo sapiens | ||
8. | ALA5200241 | 11i | IC50 | = | 17 | nM | ALA5133121 | 7.77 | nM | Homo sapiens | ||
9. | ALA5178564 | 11h | IC50 | = | 31 | nM | ALA5133121 | 7.51 | nM | Homo sapiens | ||
10. | ALA5186575 | 11g | IC50 | = | 15 | nM | ALA5133121 | 7.82 | nM | Homo sapiens | ||
11. | ALA5205781 | 11f, racemic mixture | IC50 | = | 11 | nM | ALA5133121 | 7.96 | nM | Homo sapiens | ||
12. | ALA5189461 | 11e | IC50 | = | 25 | nM | ALA5133121 | 7.60 | nM | Homo sapiens | ||
13. | ALA5195236 | 11d, racemic mixture | IC50 | = | 42 | nM | ALA5133121 | 7.38 | nM | Homo sapiens | ||
14. | ALA5207070 | 11c | IC50 | = | 39 | nM | ALA5133121 | 7.41 | nM | Homo sapiens | ||
15. | ALA5189688 | 11b | IC50 | = | 48 | nM | ALA5133121 | 7.32 | nM | Homo sapiens | ||
16. | ALA5183080 | 11a | IC50 | = | 45 | nM | ALA5133121 | 7.35 | nM | Homo sapiens | ||
17. | ALA5197788 | 10e | IC50 | = | 168 | nM | ALA5133121 | 6.78 | nM | Homo sapiens | ||
18. | ALA5197416 | 10d | IC50 | = | 483 | nM | ALA5133121 | 6.32 | nM | Homo sapiens | ||
19. | ALA5179179 | 10c | IC50 | > | 10000 | nM | ALA5133121 | nM | Homo sapiens | |||
20. | ALA5196975 | 10b | IC50 | = | 1570 | nM | ALA5133121 | 5.80 | nM | Homo sapiens |