# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA2425654 | 3 | INH | < | 50 | % | ALA2428333 | % | Homo sapiens | |||
2. | ALA2425645 | 11 | INH | < | 50 | % | ALA2428333 | % | Homo sapiens | |||
3. | ALA2425644 | 13 | INH | < | 50 | % | ALA2428333 | % | Homo sapiens | |||
4. | ALA2425646 | 12 | INH | < | 50 | % | ALA2428333 | % | Homo sapiens | |||
5. | LDN-193189 | 13 | IC50 | = | 13.3 | nM | ALA2390526 | 7.88 | nM | Homo sapiens | ||
6. | LDN 212854 | 13m | IC50 | = | 14.4 | nM | ALA2390526 | 7.84 | nM | Homo sapiens | ||
7. | ALA511563 | 52 | IC50 | = | 26.5 | nM | ALA2390526 | 7.58 | nM | Homo sapiens | ||
8. | DMH-1 | 3, DMH1, VU0364852 | IC50 | = | 27 | nM | ALA2390526 | 7.57 | nM | Homo sapiens | ||
9. | 4-[4-[3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl]phenyl]morpholine | 13a | IC50 | = | 42.1 | nM | ALA2390526 | 7.38 | nM | Homo sapiens | ||
10. | ML 347 | 50 | IC50 | = | 46 | nM | ALA2390526 | 7.34 | nM | Homo sapiens | ||
11. | ALA2385600 | 7d | IC50 | = | 52.4 | nM | ALA2390526 | 7.28 | nM | Homo sapiens | ||
12. | ALA2385586 | 13h | IC50 | = | 55 | nM | ALA2390526 | 7.26 | nM | Homo sapiens | ||
13. | Dorsomorphin | 1 | IC50 | = | 106.3 | nM | ALA2390526 | 6.97 | nM | Homo sapiens | ||
14. | 4-[4-(3-quinolin-4-ylpyrazolo[1,5-a]pyrimidin-6-yl)phenyl]morpholine | 13d | IC50 | < | 5 | nM | ALA2390526 | nM | Homo sapiens | |||
15. | 4-[6-[4-(4-methylpiperazin-1-yl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | 13r | IC50 | < | 5 | nM | ALA2390526 | nM | Homo sapiens | |||
16. | ALA2024684 | 2,PF-03671148 | IC50 | > | 5 | uM | ALA2026332 | nM | Homo sapiens | |||
17. | ALA4080797 | 35 | Activity | = | 100 | % | ALA4055149 | % | Homo sapiens | |||
18. | ALA4096145 | 2 | Activity | = | 100 | % | ALA4055149 | % | Homo sapiens | |||
19. | ALA111612 | 10a | % Control | 100 | % | ALA4879576 | Not Active | % | Homo sapiens | |||
20. | ALA4526341 | EUB0000736 | % Control | 100 | % | ALA4879576 | Not Active | % | Homo sapiens |