# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA3798256 | 6a | Activity | = | 88 | % | ALA3804402 | % | Homo sapiens | |||
2. | ALA3798574 | INK128 | IC50 | 0 | ALA3801325 | Not Determined | Homo sapiens | |||||
3. | ALA3797834 | 18 | IC50 | = | 137 | nM | ALA3801325 | 6.86 | nM | Homo sapiens | ||
4. | ALA3797933 | 17 | IC50 | = | 4.7 | nM | ALA3801325 | 8.33 | nM | Homo sapiens | ||
5. | eCF309 | 12 | INH | = | 77 | % | ALA3803014 | % | Homo sapiens | |||
6. | eCF309 | 12 | IC50 | = | 2110 | nM | ALA3801325 | 5.68 | nM | Homo sapiens | ||
7. | ALA3780219 | 18a | Activity | = | 0 | % | ALA3784719 | % | Homo sapiens | |||
8. | Dasatinib | 2, BMS-354825 | GI50 | = | 3 | uM | ALA3784003 | nM | Homo sapiens | |||
9. | Nilotinib (AMN-107) | 38 | GI50 | = | 1.1 | uM | ALA3784003 | nM | Homo sapiens | |||
10. | Imatinib (STI571) | 1 | GI50 | = | 3 | uM | ALA3784003 | nM | Homo sapiens | |||
11. | ALA3780219 | 18a | GI50 | = | 3.3 | uM | ALA3784003 | nM | Homo sapiens | |||
12. | ALA3780219 | 18a | IC50 | = | 292 | nM | ALA3783996 | 6.54 | nM | Homo sapiens | ||
13. | ALA3758502 | 1 | INH | = | 52.6 | % | ALA3762328 | % | Homo sapiens | |||
14. | ALA3745885 | 7ao; ON1231320 | IC50 | > | 10 | uM | ALA3749003 | nM | Homo sapiens | |||
15. | ALA3747489 | 21 | INH | = | 85 | % | ALA3750791 | % | Homo sapiens | |||
16. | ALA3746293 | 23 | INH | = | 0.8 | % | ALA3751093 | % | Homo sapiens | |||
17. | ALA3745857 | 47 | INH | = | 51 | % | ALA3750646 | % | Homo sapiens | |||
18. | ALA3746973 | 41 | INH | = | 99 | % | ALA3750646 | % | Homo sapiens | |||
19. | ALA3746951 | 40 | INH | = | 95 | % | ALA3750646 | % | Homo sapiens | |||
20. | ALA3747023 | 29 | INH | = | 89 | % | ALA3750646 | % | Homo sapiens |